Design, synthesis, and evaluation in vitro of quinoline-8-carboxamides, a new class of poly (adenosine-diphosphate-ribose) polymerase-1 (PARP-1) inhibitor

AM Lord, MF Mahon, MD Lloyd…

Index: Journal of Medicinal Chemistry, , vol. 52, # 3 p. 868 - 877

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Citation Number: 50

Abstract

... Journal of Medicinal Chemistry. ... To whom correspondence should be addressed. Telephone: +44 1225 386840. Fax: +44 1225 386114. E-mail: mdthreadgill@bath.ac.uk., † Department of Pharmacy and Pharmacology. , ‡ Department of Chemistry. ...