Synthesis and Biological Evaluation of Metabolites of 2-n-Butyl-9-methyl-8-[1, 2, 3] triazol-2-yl-9 H-purin-6-ylamine (ST1535), A Potent Antagonist of the A2A …

…, T Riccioni, F Borsini, G Tarzia, P Minetti

Index: Kotek, Vladislav; Chudikova, Nadezda; Tobrman, Tomas; Dvorak, Dalimil Organic Letters, 2010 , vol. 12, # 24 p. 5724 - 5727

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Citation Number: 13

Abstract

... Volume: Page: ... 2013, 56 (13), pp 5456–5463. DOI: 10.1021/jm400491x. Publication Date (Web): June 12, 2013. Copyright ... methyl-8-(2H-1,2,3-triazol-2-yl)-9H-purines is based on the general I–Mg exchange reaction of 2,6-dihalopurines proposed by Dvořák(7) to ...