Structure–activity relationships of diamine inhibitors of cytochrome P450 (CYP) 3A as novel pharmacoenhancers. Part II: P2/P3 region and discovery of cobicistat (GS- …

L Xu, H Liu, A Hong, R Vivian, BP Murray…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 24, # 3 p. 995 - 999

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Citation Number: 8

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... a Department of Medicinal Chemistry, Gilead Sciences ... e Department of Structural Chemistry, Gilead Sciences, 333 Lakeside Drive, Foster City, CA 94303, USA. Received 13 November 2013, Revised 10 December 2013, Accepted 11 ...