Tetrahedron Letters

Straightforward synthesis of orthogonally protected piperidin-3-ylmethanamine and piperidin-4-ylmethanamine derivatives

U Košak, B Brus, S Gobec

Index: Kosak, Urban; Brus, Boris; Gobec, Stanislav Tetrahedron Letters, 2014 , vol. 55, # 12 p. 2037 - 2039

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Citation Number: 5

Abstract

Abstract The 1, 3-and 1, 4-disubstituted piperidines are important building blocks in medicinal chemistry and drug discovery. We present the synthesis of orthogonally protected piperidin-3-ylmethanamine and piperidin-4-ylmethanamine derivatives from commercially ...