Synthesis and biological evaluation of 3-[4-(amino/methylsulfonyl) phenyl] methylene-indolin-2-one derivatives as novel COX-1/2 and 5-LOX inhibitors

Y Lai, L Ma, W Huang, X Yu, Y Zhang, H Ji…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 20, # 24 p. 7349 - 7353

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Citation Number: 29

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... b Department of Pharmacology, China Pharmaceutical University, Nanjing 210009, PR China; c Department of Molecular and Medical Pharmacology, University of California Los Angeles, Los Angeles, CA 90095, USA. ...