Oxidative Biaryl Coupling of Thiophenes and Thiazoles with Arylboronic Acids through Palladium Catalysis: Otherwise Difficult C4??Selective C H Arylation Enabled …

S Kirchberg, S Tani, K Ueda…

Index: Waki, Minoru; Maegawa, Yoshifumi; Hara, Kenji; Goto, Yasutomo; Shirai, Soichi; Yamada, Yuri; Mizoshita, Norihiro; Tani, Takao; Chun, Wang-Jae; Muratsugu, Satoshi; Tada, Mizuki; Fukuoka, Atsushi; Inagaki, Shinji Journal of the American Chemical Society, 2014 , vol. 136, # 10 p. 4003 - 4011

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Citation Number: 134

Abstract

Heteroarenes equipped with aryl groups (heterobiaryls) are often found in biologically active compounds, organic materials, and pharmaceuticals. In recent years, the direct CÀH arylation of heteroarenes catalyzed by a transition-metal complex [1, 2] has emerged as a