Synlett

Desulfonylation of Indoles and 7-Azaindoles Using Sodium tert-Butoxide

…, C Croix, J Basset, MD Pujol, MC Viaud-Massuard

Index: Chaulet, Charlotte; Croix, Cecile; Basset, Joan; Pujol, Maria-Dolores; Viaud-Massuard, Marie-Claude Synlett, 2010 , # 10 p. 1481 - 1484

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Citation Number: 5

Abstract

Abstract A mild method for the desulfonylation of N-indoles and N-azaindoles is described. Deprotection is carried out under basic conditions, using sodium tert-butoxide in dioxane. Several functionalized indoles and 7-azaindoles were efficiently deprotected by this ...

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