Tetrahedron

Nickel-catalysed couplings of aryl chlorides with secondary amines and piperazines

E Brenner, R Schneider, Y Fort

Index: Brenner, Eric; Schneider, Raphael; Fort, Yves Tetrahedron, 1999 , vol. 55, # 44 p. 12829 - 12842

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Citation Number: 109

Abstract

Abstract: The reaction of aryl chlorides with secondary amines or piperazines in the presence of an in situ generated liganded nickel catalyst gives arylamines in good yields. Our process provides a mild, convenient and cheap method of arylamination starting from readily available substlates.© 1999 Elsevier Science Ltd. All rights reserved.

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