e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Efficient one-step synthesis of trialkylsubstituted 2 (5H)-furanones utilizing direct Ti-crossed aldol condensation and its application to the straightforward synthesis of ( …
TiCl4–Bu3N-mediated condensation of ketones with α, α-dimethoxyketones afforded trialkylsubstituted 2 (5H)-furanones in a one-pot manner, wherein aldol addition and furanone formation occurred sequentially; its application to straightforward synthesis of (R)- mintlactone and (R)-menthofuran, two representative natural mint perfumes, is demonstrated.