e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Preparation of and Fluoroalkylation with (Chlorodifluoromethyl) trimethylsilane, Difluorobis (trimethylsilyl) methane, and 1, 1, 2, 2-Tetrafluoro-1, 2-bis (trimethylsilyl) …
…, D Deffieux, M Bradley, R Bau, GA Olah
Index: Yudin, Andrei K.; Prakash, G. K. Surya; Deffieux, Denis; Bradley, Michael; Bau, Robert; Olah, George A. Journal of the American Chemical Society, 1997 , vol. 119, # 7 p. 1572 - 1581
CF2BrCl reacts with aluminum/N-methylpyrrolidinone in the presence of chlorotrimethylsilane to give Me3SiCF2Cl in high yield. Similarly, CF2Br2 gives Me3SiCF2Br with bromotrimethylsilane. Chlorodifluoromethylation of aldehydes using Me3SiCF2Cl and a catalytic amount of TBAF in polar solvents occurs at room temperature, providing difluoromethylated alcohols in two steps. Electroreduction of Me3SiCF2Cl in the presence ...