Preparation of (S)-piperazine-2-carboxylic acid,(R)-piperazi...
[Eichhorn, Eric; Roduit, Jean-Paul; Shaw, Nicholas; Heinzmann, Klaus; Kiener, Andreas Tetrahedron Asymmetry, 1997 , vol. 8, # 15 p. 2533 - 2536]
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Design and synthesis of peripherally restricted transient re...
[Tamayo, Nuria; Liao, Hongyu; Stec, Markian M.; Wang, Xianghong; Chakrabarti, Partha; Retz, Dan; Doherty, Elizabeth M.; Surapaneni, Sekhar; Tamir, Rami; Bannon, Anthony W.; Gavva, Narender R.; Norman, Mark H. Journal of Medicinal Chemistry, 2008 , vol. 51, # 9 p. 2744 - 2757]
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Core refinement toward permeable β-secretase (BACE-1) inhibi...
[Ginman, Tobias; Viklund, Jenny; Malmstroem, Jonas; Blid, Jan; Emond, Rikard; Forsblom, Rickard; Johansson, Anh; Kers, Annika; Lake, Fredrik; Sehgelmeble, Fernando; Sterky, Karin J.; Bergh, Margareta; Lindgren, Anders; Johansson, Patrik; Jeppsson, Fredrik; Faelting, Johanna; Gravenfors, Ylva; Rahm, Fredrik Journal of Medicinal Chemistry, 2013 , vol. 56, # 11 p. 4181 - 4205]
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Oxidation of secondary amines to α-cyanoamines
[Tetrahedron Letters, , vol. 26, # 9 p. 1229 - 1232]
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Oxidation of secondary amines to α-cyanoamines
[Tetrahedron Letters, , vol. 26, # 9 p. 1229 - 1232]
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