Practical asymmetric synthesis of efavirenz (DMP 266), an HIV-1 reverse transcriptase inhibitor

ME Pierce, RL Parsons, LA Radesca…

Index: Journal of Organic Chemistry, , vol. 63, # 23 p. 8536 - 8543

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Citation Number: 179

Abstract

... The Journal of Organic Chemistry. ... Department of Process Research, Merck Research Laboratories, PO Box 2000, Rahway, New Jersey 07065. J. Org. Chem. , 1998, 63 (23), pp 8536–8543. DOI: 10.1021/jo981170l. Publication ...

Practical asymmetric synthesis of efavirenz (DMP 266), an HI...

[Pierce, Michael E.; Parsons Jr., Rodney L.; Radesca, Lilian A.; Lo, Young S.; Silverman, Stuart; Moore, James R.; Islam, Qamrul; Choudhury, Anusuya; Fortunak, Joseph M. D.; Nguyen, Dieu; Luo, Chi; Morgan, Susan J.; Davis, Wayne P.; Confalone, Pat N.; Chen, Cheng-Yi; Tillyer, Richard D.; Frey, Lisa; Tan, Lushi; Xu, Feng; Zhao, Dalian; Thompson, Andrew S.; Corley, Edward G.; Grabowski, Edward J. J.; Reamer, Robert; Reider, Paul J. Journal of Organic Chemistry, 1998 , vol. 63, # 23 p. 8536 - 8543]

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