Solid-phase synthesis of 1, 4-benzodiazepine-2, 5-diones. Library preparation and demonstration of synthesis generality

CG Boojamra, KM Burow, LA Thompson…

Index: Akssira; Boumzebra; Kasmi; Dahdouh; Roumestant; Viallefont Synthetic Communications, 1993 , vol. 23, # 16 p. 2265 - 2272

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Citation Number: 211

Abstract

... Volume: Page: ... 1d was cleaved from support, an aliquot of resin was subjected to cross-coupling with p-methoxybenzeneboronic acid ... The library was prepared predominantly to demonstrate that our synthetic method proceeds with high fidelity, even when ...