Antagonists of the human A2A adenosine receptor. 4. Design, synthesis, and preclinical evaluation of 7-aryltriazolo [4, 5-d] pyrimidines

RJ Gillespie, SJ Bamford, R Botting…

Index: Journal of Medicinal Chemistry, , vol. 52, # 1 p. 33 - 47

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Citation Number: 67

Abstract

... Journal of Medicinal Chemistry. ... These issues clearly highlight the urgent medical need for an alternative point of therapeutic intervention that can alleviate the symptoms of the disease while additionally offering predictable pharmacokinetics and a reduced incidence of side ...

Supramolecular complexes obtained from porphyrin–crown ether...

[Solladie, Nathalie; Walther, Mathieu E.; Herschbach, Haiko; Leize, Emmanuelle; Dorsselaer, Alain Van; Duarte, Teresa M. Figueira; Nierengarten, Jean-Francois Tetrahedron, 2006 , vol. 62, # 9 p. 1979 - 1987]

Development of irreversible diphenyl phosphonate inhibitors ...

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Design, synthesis, and proposed active site binding analysis...

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A supramolecular oligophenylenevinylene–C 60 conjugate

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