Tetrahedron Letters

Microwave-assisted Sonogashira-type cross couplings of various heterocyclic methylthioethers

BC Shook, D Chakravarty, PF Jackson

Index: Shook, Brian C.; Chakravarty, Devraj; Jackson, Paul F. Tetrahedron Letters, 2009 , vol. 50, # 9 p. 1013 - 1015

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Citation Number: 22

Abstract

A novel, microwave-assisted, palladium-catalyzed Sonogashira-type coupling of terminal alkynes with a variety of heteroaryl thiomethylethers is reported. The developed protocol allows for further utility and diversification of a number of chemically and biologically interesting scaffolds.

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