Rapid preparation of triazolyl substituted NH-heterocyclic kinase inhibitors via one-pot Sonogashira coupling–TMS-deprotection–CuAAC sequence

E Merkul, F Klukas, D Dorsch, U Grädler…

Index: Organic and Biomolecular Chemistry, , vol. 9, # 14 p. 5129 - 5136

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Citation Number: 26

Abstract

... Chem., 2011, 9, 5129-5136 Show Compounds Show Chemical Terms Show ... dihydro)pyrazine (dragmacidins, 7 hamacanthins 8 ), oxazinone (oxazinins 9 ), oxadiazinone (alboinon ... has attracted considerable attention in bioconjugate chemistry, medicinal chemistry, and drug ...