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KYT-1

更新时间:2025-08-25 15:34:32

KYT-1结构式
KYT-1结构式
委托求购
常用名 KYT-1 英文名 KYT-1
CAS号 241825-16-1 分子量 619.768
密度 N/A 沸点 N/A
分子式 C29H49N9O6 熔点 N/A
MSDS N/A 闪点 N/A

 KYT-1用途


KYT-1是一种有效、选择性的牙龈假单胞菌毒力因子Arg-gingipain(Rgp)抑制剂,Ki为40 nM(RgpA/B)。KYT-1对牙龈卟啉单胞菌刺激的SMC增殖有明显的抑制作用。

 KYT-1名称

英文名 KYT-1

 KYT-1生物活性

描述 KYT-1是一种有效、选择性的牙龈假单胞菌毒力因子Arg-gingipain(Rgp)抑制剂,Ki为40 nM(RgpA/B)。KYT-1对牙龈卟啉单胞菌刺激的SMC增殖有明显的抑制作用。
参考文献 1. Kadowaki T, et al. Mol Pharmacol. 2004 Dec;66(6):1599-606. 2. Hosn KN, et al. Clin Exp Dent Res. 2015 Oct 27;1(1):18-25. 3. Inaba H, et al. J Periodontol. 2011 Nov;82(11):1616-22. 4. Cao C, et al. Int J Clin Exp Med. 2015 Oct 15;8(10):18327-34.

 KYT-1物理化学性质

分子式 C29H49N9O6
分子量 619.768
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