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AGH-107

更新时间:2024-04-05 18:05:12

AGH-107结构式
AGH-107结构式
委托求购
常用名 AGH-107 英文名 AGH-107
CAS号 2172907-10-5 分子量 337.164
密度 N/A 沸点 N/A
分子式 C13H12In3 熔点 N/A
MSDS N/A 闪点 N/A

 AGH-107用途


AGH-107是一种有效、选择性的5-HT7受体激动剂,Ki为6 nM,EC50为19 nM,选择性是5-HT1AR的176倍。AGH-107在HEK-293和HepG2细胞培养中表现出对相关CNS靶点的高选择性、高代谢稳定性和低毒性。

 AGH-107名称

英文名 AGH-107

 AGH-107生物活性

描述 AGH-107是一种有效、选择性的5-HT7受体激动剂,Ki为6 nM,EC50为19 nM,选择性是5-HT1AR的176倍。AGH-107在HEK-293和HepG2细胞培养中表现出对相关CNS靶点的高选择性、高代谢稳定性和低毒性。
参考文献 1. Hogendorf AS, et al. Sci Rep. 2017 May 4;7(1):1444.

 AGH-107物理化学性质

分子式 C13H12In3
分子量 337.164
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