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983-80-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:P388
External ID: CHEMBL762217
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1987
Volume: 30
Issue: 12
First Page: 2181
Last Page: 2190
DOI: 10.1021/jm00395a004

Target ChEMBL ID: CHEMBL389
ChEMBL Target Name: P388
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
ILSmax=35
ILSmax=80
ILSmax=107
ILSmax=80
ILSmax=51
ILSmax=40
ILSmax=70
ILSmax=50
ILSmax=38
ILSmax=60
ILSmax=35
ILSmax=86
ILSmax=60
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL723207
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1987
Volume: 30
Issue: 12
First Page: 2181
Last Page: 2190
DOI: 10.1021/jm00395a004

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MTD=95uM kg-1
MTD=60uM kg-1
MTD=50uM kg-1
MTD=60uM kg-1
MTD=320uM kg-1
MTD=300uM kg-1
MTD=110uM kg-1
MTD=670uM kg-1
MTD=320uM kg-1
MTD=120uM kg-1
MTD=72uM kg-1
MTD>600uM kg-1
MTD=280uM kg-1
MTD=18uM kg-1
MTD=48uM kg-1
MTD=82uM kg-1
MTD>300uM kg-1
MTD=1000uM kg-1
MTD=17uM kg-1
MTD=80uM kg-1