前往化源商城

96889-94-0 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Proteus vulgaris
External ID: CHEMBL831511
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL614450
ChEMBL Target Name: Proteus vulgaris
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=50ug.mL-1
MIC=100ug.mL-1
MIC=50ug.mL-1
MIC=50ug.mL-1
MIC=25ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium sp.
External ID: CHEMBL5262816
Protocol: N/A
Comment: Journal: Eur J Med Chem
Year: 2017
Volume: 137
First Page: 504
Last Page: 544
DOI: 10.1016/j.ejmech.2017.06.005

Target ChEMBL ID: CHEMBL612963
ChEMBL Target Name: Mycobacterium sp.
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=1.56ug.mL-1
MIC=12.5ug.mL-1
MIC=0.78ug.mL-1
MIC<100ug.mL-1
MIC=128ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Raji
External ID: CHEMBL1018461
Protocol: N/A
Comment: Journal: J. Nat. Prod.
Year: 1989
Volume: 52
Issue: 5
First Page: 987
Last Page: 995
DOI: 10.1021/np50065a012

Target ChEMBL ID: CHEMBL614628
ChEMBL Target Name: Raji
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity=70%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL830605
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=25ug.mL-1
MIC>100ug.mL-1
MIC=6.25ug.mL-1
MIC=12.5ug.mL-1
MIC=1.56ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium intracellulare
External ID: CHEMBL751965
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1992
Volume: 35
Issue: 22
First Page: 4069
Last Page: 4077
DOI: 10.1021/jm00100a012

Target ChEMBL ID: CHEMBL612640
ChEMBL Target Name: Mycobacterium intracellulare
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=1.56ug.mL-1
MIC=12.5ug.mL-1
MIC=1.56ug.mL-1
MIC=0.78ug.mL-1
MIC=0.39ug.mL-1
MIC=0.78ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Aspergillus fumigatus
External ID: CHEMBL648395
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1992
Volume: 35
Issue: 22
First Page: 4069
Last Page: 4077
DOI: 10.1021/jm00100a012

Target ChEMBL ID: CHEMBL363
ChEMBL Target Name: Aspergillus fumigatus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=0.39ug.mL-1
MIC=100ug.mL-1
MIC=1.56ug.mL-1
MIC=0.39ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL830617
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=50ug.mL-1
MIC=100ug.mL-1
MIC=6.25ug.mL-1
MIC=6.25ug.mL-1
MIC=3.13ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium intracellulare
External ID: CHEMBL2438881
Protocol: N/A
Comment: Journal: Eur J Med Chem
Year: 2013
Volume: 67
First Page: 98
Last Page: 110
DOI: 10.1016/j.ejmech.2013.06.010

Target ChEMBL ID: CHEMBL612640
ChEMBL Target Name: Mycobacterium intracellulare
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=12.5ug.mL-1
MIC=0.78ug.mL-1
MIC=0.39ug.mL-1
MIC=0.5ug.mL-1
MIC=2ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Bacillus subtilis
External ID: CHEMBL875742
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL359
ChEMBL Target Name: Bacillus subtilis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=25ug.mL-1
MIC=100ug.mL-1
MIC=3.13ug.mL-1
MIC=6.25ug.mL-1
MIC=3.13ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4629203
Protocol: N/A
Comment: Journal: Bioorg Med Chem
Year: 2020
Volume: 28
Issue: 10
First Page: 115462
Last Page: 115462
DOI: 10.1016/j.bmc.2020.115462
PubChem Standard ValueStandard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
154.5IC50=154500nMOutside typical range
83.5IC50=83500nM
11.3IC50=11300nM
57.9IC50=57900nM
38.3IC50=38300nM
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Aspergillus niger
External ID: CHEMBL831782
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL358
ChEMBL Target Name: Aspergillus niger
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=100ug.mL-1
MIC=100ug.mL-1
MIC=12.5ug.mL-1
MIC=12.5ug.mL-1
MIC=3.13ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mucor mucedo
External ID: CHEMBL875738
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL613767
ChEMBL Target Name: Mucor mucedo
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=50ug.mL-1
MIC>100ug.mL-1
MIC=6.25ug.mL-1
MIC=12.5ug.mL-1
MIC=3.13ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Rhodotorula mucilaginosa
External ID: CHEMBL831783
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL612871
ChEMBL Target Name: Rhodotorula mucilaginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=50ug.mL-1
MIC=100ug.mL-1
MIC=6.25ug.mL-1
MIC=12.5ug.mL-1
MIC=3.13ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:NON-PROTEIN TARGET
External ID: CHEMBL1005708
Protocol: N/A
Comment: Journal: J. Nat. Prod.
Year: 2001
Volume: 64
Issue: 5
First Page: 616
Last Page: 619
DOI: 10.1021/np0005208

Target ChEMBL ID: CHEMBL3879801
ChEMBL Target Name: NON-PROTEIN TARGET
ChEMBL Target Type: NON-MOLECULAR - Target has not been defined at a molecular level, only the non-molecular entity which is affected (e.g., organism, cell line etc)
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
IC50=0.54ug.mL-1
IC50=1.9ug.mL-1
IC50=2.4ug.mL-1
IC50=3.8ug.mL-1
IC50=0.36ug.mL-1
IC50=10.6ug.mL-1
IC50=0.01ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL5128127
Protocol: N/A
Comment: Journal: Eur J Med Chem
Year: 2022
Volume: 232
First Page: 114173
Last Page: 114173
DOI: 10.1016/j.ejmech.2022.114173

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=6.25ug.mL-1
MIC=12.5ug.mL-1
MIC=12.5ug.mL-1
MIC=16ug.mL-1
MIC=16ug.mL-1
MIC=12.5ug.mL-1
MIC=12.5ug.mL-1
MIC=12.5ug.mL-1
MIC=12.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:NON-PROTEIN TARGET
External ID: CHEMBL831447
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL3879801
ChEMBL Target Name: NON-PROTEIN TARGET
ChEMBL Target Type: NON-MOLECULAR - Target has not been defined at a molecular level, only the non-molecular entity which is affected (e.g., organism, cell line etc)
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=50ug.mL-1
MIC=50ug.mL-1
MIC=3.13ug.mL-1
MIC=12.5ug.mL-1
MIC=1.56ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:HepG2
External ID: CHEMBL1005707
Protocol: N/A
Comment: Journal: J. Nat. Prod.
Year: 2001
Volume: 64
Issue: 5
First Page: 616
Last Page: 619
DOI: 10.1021/np0005208

Target ChEMBL ID: CHEMBL395
ChEMBL Target Name: HepG2
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
IC50=0.22ug.mL-1
IC50=6.6ug.mL-1
IC50=6.2ug.mL-1
IC50=0.22ug.mL-1
IC50=0.01ug.mL-1
IC50=3.9ug.mL-1
IC50=1.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Candida albicans
External ID: CHEMBL654185
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1992
Volume: 35
Issue: 22
First Page: 4069
Last Page: 4077
DOI: 10.1021/jm00100a012

Target ChEMBL ID: CHEMBL366
ChEMBL Target Name: Candida albicans
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=0.78ug.mL-1
MIC=1.56ug.mL-1
MIC=12.5ug.mL-1
MIC=25ug.mL-1
MIC=1.56ug.mL-1
MIC=0.39ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Saccharomyces cerevisiae
External ID: CHEMBL830691
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL361
ChEMBL Target Name: Saccharomyces cerevisiae
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=100ug.mL-1
MIC=100ug.mL-1
MIC=12.5ug.mL-1
MIC=25ug.mL-1
MIC=3.13ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Rhizopus microsporus var. chinensis
External ID: CHEMBL831798
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL612840
ChEMBL Target Name: Rhizopus microsporus var. chinensis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>100ug.mL-1
MIC>100ug.mL-1
MIC=12.5ug.mL-1
MIC=25ug.mL-1
MIC=12.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Cyberlindnera jadinii
External ID: CHEMBL831412
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL612309
ChEMBL Target Name: Cyberlindnera jadinii
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=50ug.mL-1
MIC=100ug.mL-1
MIC=12.5ug.mL-1
MIC=25ug.mL-1
MIC=12.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Raji
External ID: CHEMBL1018458
Protocol: N/A
Comment: Journal: J. Nat. Prod.
Year: 1989
Volume: 52
Issue: 5
First Page: 987
Last Page: 995
DOI: 10.1021/np50065a012

Target ChEMBL ID: CHEMBL614628
ChEMBL Target Name: Raji
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity=0%
Activity=20%
Activity=70%
Activity=0%
Activity=40%
Activity>80%
Activity=40%
Activity>80%
Activity=60%
Activity>80%
Activity=70%
Activity>80%
Activity=20%
Activity=70%
Activity=0%
Activity=0%
Activity=0%
Activity=70%
Activity>80%
Activity=70%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL1018457
Protocol: N/A
Comment: Journal: J Nat Prod
Year: 1989
Volume: 52
Issue: 5
First Page: 987
Last Page: 995
DOI: 10.1021/np50065a012
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=31.5%
Inhibition=68.9%
Inhibition=100%
Inhibition=89.4%
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=89.2%
Inhibition=100%
Inhibition=94.2%
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=32.7%
Inhibition=59.4%
Inhibition=81.4%
Inhibition=100%
Inhibition=100%
Inhibition=100%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Raji
External ID: CHEMBL1018460
Protocol: N/A
Comment: Journal: J. Nat. Prod.
Year: 1989
Volume: 52
Issue: 5
First Page: 987
Last Page: 995
DOI: 10.1021/np50065a012

Target ChEMBL ID: CHEMBL614628
ChEMBL Target Name: Raji
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity=50%
Activity=50%
Activity>80%
Activity=70%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity=50%
Activity>80%
Activity=70%
Activity=10%
Activity=70%
Activity>80%
Activity>80%
Activity>80%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Raji
External ID: CHEMBL1018459
Protocol: N/A
Comment: Journal: J. Nat. Prod.
Year: 1989
Volume: 52
Issue: 5
First Page: 987
Last Page: 995
DOI: 10.1021/np50065a012

Target ChEMBL ID: CHEMBL614628
ChEMBL Target Name: Raji
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity=10%
Activity=40%
Activity>80%
Activity=0%
Activity=60%
Activity>80%
Activity=60%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity>80%
Activity=50%
Activity>80%
Activity=0%
Activity=10%
Activity=0%
Activity>80%
Activity>80%
Activity>80%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL831422
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>100ug.mL-1
MIC>100ug.mL-1
MIC>100ug.mL-1
MIC>100ug.mL-1
MIC>100ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL1015774
Protocol: N/A
Comment: Journal: J Nat Prod
Year: 1989
Volume: 52
Issue: 5
First Page: 987
Last Page: 995
DOI: 10.1021/np50065a012
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=0%
Inhibition=0%
Inhibition=89.5%
Inhibition=0%
Inhibition=0%
Inhibition=18.2%
Inhibition=0%
Inhibition=0%
Inhibition=71.4%
Inhibition=23.8%
Inhibition=27.1%
Inhibition=28.5%
Inhibition=0%
Inhibition=34.6%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=40.6%
Inhibition=45.8%
Inhibition=55.5%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL1018456
Protocol: N/A
Comment: Journal: J Nat Prod
Year: 1989
Volume: 52
Issue: 5
First Page: 987
Last Page: 995
DOI: 10.1021/np50065a012
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=15.8%
Inhibition=0%
Inhibition=100%
Inhibition=65.7%
Inhibition=88.4%
Inhibition=91.1%
Inhibition=97.8%
Inhibition=61.5%
Inhibition=100%
Inhibition=71.2%
Inhibition=92.3%
Inhibition=89.9%
Inhibition=37.5%
Inhibition=100%
Inhibition=0%
Inhibition=0%
Inhibition=52.8%
Inhibition=77.5%
Inhibition=92.5%
Inhibition=100%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Cryptococcus neoformans
External ID: CHEMBL660674
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1992
Volume: 35
Issue: 22
First Page: 4069
Last Page: 4077
DOI: 10.1021/jm00100a012

Target ChEMBL ID: CHEMBL365
ChEMBL Target Name: Cryptococcus neoformans
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=0.39ug.mL-1
MIC=0.78ug.mL-1
MIC=1.56ug.mL-1
MIC=25ug.mL-1
MIC=0.78ug.mL-1
MIC=1.56ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL1015775
Protocol: N/A
Comment: Journal: J Nat Prod
Year: 1989
Volume: 52
Issue: 5
First Page: 987
Last Page: 995
DOI: 10.1021/np50065a012
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=0%
Inhibition=0%
Inhibition=100%
Inhibition=0%
Inhibition=0%
Inhibition=54.2%
Inhibition=13.1%
Inhibition=60.5%
Inhibition=92.4%
Inhibition=61.9%
Inhibition=70.1%
Inhibition=78.6%
Inhibition=0%
Inhibition=54.3%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=48.7%
Inhibition=89.2%
Inhibition=94.1%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Schizosaccharomyces pombe
External ID: CHEMBL830701
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2005
Volume: 15
Issue: 4
First Page: 1079
Last Page: 1082
DOI: 10.1016/j.bmcl.2004.12.059

Target ChEMBL ID: CHEMBL612632
ChEMBL Target Name: Schizosaccharomyces pombe
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=25ug.mL-1
MIC=50ug.mL-1
MIC=3.13ug.mL-1
MIC=1.56ug.mL-1
MIC=0.78ug.mL-1