前往化源商城

921908-34-1 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Onchocerca ochengi
External ID: CHEMBL2093846
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL2093135
ChEMBL Target Name: Onchocerca ochengi
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: WHO Tropical Disease Research (TDR) Malaria Screening
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=60%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=100%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Onchocerca ochengi
External ID: CHEMBL2093845
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL2093135
ChEMBL Target Name: Onchocerca ochengi
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: WHO Tropical Disease Research (TDR) Malaria Screening
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=0%
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=100%
Inhibition=0%
Inhibition=100%
Inhibition=100%
Inhibition=0%
Inhibition=50%
Inhibition=100%
Inhibition=50%
Inhibition=100%
Inhibition=0%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Trypanosoma cruzi
External ID: CHEMBL2093838
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL368
ChEMBL Target Name: Trypanosoma cruzi
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: WHO Tropical Disease Research (TDR) Malaria Screening
Standard TypeStandard RelationStandard ValueStandard Units
IC50>11.76ug.mL-1
IC503.282ug.mL-1
IC503.303ug.mL-1
IC50=0.305ug.mL-1
IC50>8.92ug.mL-1
IC50>12.94ug.mL-1
IC50=4.255ug.mL-1
IC50=5.134ug.mL-1
IC50>13.07ug.mL-1
IC50=2.928ug.mL-1
IC50>10.72ug.mL-1
IC50=0.398ug.mL-1
IC50=0.511ug.mL-1
IC50=0.345ug.mL-1
IC50=0.929ug.mL-1
IC50=5.242ug.mL-1
IC50=5.157ug.mL-1
IC503.089ug.mL-1
IC50=0.575ug.mL-1
IC50=0.442ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Trypanosoma brucei brucei
External ID: CHEMBL2093839
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL612851
ChEMBL Target Name: Trypanosoma brucei brucei
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: WHO Tropical Disease Research (TDR) Malaria Screening
Standard TypeStandard RelationStandard ValueStandard Units
IC50>11.76ug.mL-1
IC50>5.735ug.mL-1
IC502.534ug.mL-1
IC50=3.231ug.mL-1
IC50>8.92ug.mL-1
IC50>12.94ug.mL-1
IC50=5.005ug.mL-1
IC50>11.95ug.mL-1
IC50>13.07ug.mL-1
IC50=3.56ug.mL-1
IC50=0.422ug.mL-1
IC50=0.292ug.mL-1
IC50=4.55ug.mL-1
IC50=0.152ug.mL-1
IC50=4.804ug.mL-1
IC50>10.99ug.mL-1
IC50=3.689ug.mL-1
IC503.135ug.mL-1
IC50>12.39ug.mL-1
IC50=4.317ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:MRC5
External ID: CHEMBL2093836
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL614181
ChEMBL Target Name: MRC5
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: WHO Tropical Disease Research (TDR) Malaria Screening
Standard TypeStandard RelationStandard ValueStandard Units
IC50>11.76ug.mL-1
IC501.813ug.mL-1
IC503.012ug.mL-1
IC50=2.04ug.mL-1
IC50>8.92ug.mL-1
IC50>12.94ug.mL-1
IC50>13.12ug.mL-1
IC50>11.95ug.mL-1
IC50>13.07ug.mL-1
IC50>11ug.mL-1
IC50>10.72ug.mL-1
IC50=1.312ug.mL-1
IC50=5.889ug.mL-1
IC50>9.013ug.mL-1
IC50>14.84ug.mL-1
IC50>10.99ug.mL-1
IC50>9.821ug.mL-1
IC501.955ug.mL-1
IC50=1.527ug.mL-1
IC50=6.19ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Plasmodium falciparum K1
External ID: CHEMBL2093837
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL612856
ChEMBL Target Name: Plasmodium falciparum K1
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: WHO Tropical Disease Research (TDR) Malaria Screening
Standard TypeStandard RelationStandard ValueStandard Units
IC50=0.24ug.mL-1
IC50>5.735ug.mL-1
IC500.566ug.mL-1
IC50=9.025ug.mL-1
IC50>8.92ug.mL-1
IC50>12.94ug.mL-1
IC50>13.12ug.mL-1
IC50>11.95ug.mL-1
IC50>13.07ug.mL-1
IC50>11ug.mL-1
IC50>10.72ug.mL-1
IC50=8.258ug.mL-1
IC50=10.23ug.mL-1
IC50>9.013ug.mL-1
IC50=0.7798ug.mL-1
IC50=7.351ug.mL-1
IC50=4.264ug.mL-1
IC50>9.912ug.mL-1
IC50>12.39ug.mL-1
IC50>13.34ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Leishmania infantum
External ID: CHEMBL2093840
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL612848
ChEMBL Target Name: Leishmania infantum
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: WHO Tropical Disease Research (TDR) Malaria Screening
Standard TypeStandard RelationStandard ValueStandard Units
IC50>11.76ug.mL-1
IC50>5.735ug.mL-1
IC50>9.19ug.mL-1
IC50=3.714ug.mL-1
IC50>8.92ug.mL-1
IC50>12.94ug.mL-1
IC50>13.12ug.mL-1
IC50>11.95ug.mL-1
IC50=4.231ug.mL-1
IC50>11ug.mL-1
IC50>10.72ug.mL-1
IC50=3.737ug.mL-1
IC50=9.575ug.mL-1
IC50>9.013ug.mL-1
IC50>14.84ug.mL-1
IC50>10.99ug.mL-1
IC50>9.821ug.mL-1
IC503.209ug.mL-1
IC50=4.011ug.mL-1
IC50=4.317ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Schistosoma mansoni
External ID: CHEMBL2093841
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL612893
ChEMBL Target Name: Schistosoma mansoni
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: WHO Tropical Disease Research (TDR) Malaria Screening
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=25%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%