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90296-07-4 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL634599
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1984
Volume: 27
Issue: 8
First Page: 967
Last Page: 978
DOI: 10.1021/jm00374a006
Standard TypeStandard RelationStandard Value
Solubility ratio=1.234
Solubility ratio=1.32
Solubility ratio=1.398
Solubility ratio=1.302
Solubility ratio=1.198
Solubility ratio=1.178
Solubility ratio=1.296
Solubility ratio=1.149
Solubility ratio=1.36
Solubility ratio=1.317
Solubility ratio=1.351
Solubility ratio=1.144
Solubility ratio=1.313
Solubility ratio=1.176
Solubility ratio=1.284
Solubility ratio=1.246
Solubility ratio=1.223
Solubility ratio=1.092
Solubility ratio=1.135
Solubility ratio=1.39
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL634600
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1984
Volume: 27
Issue: 8
First Page: 967
Last Page: 978
DOI: 10.1021/jm00374a006
Standard TypeStandard RelationStandard ValueActivity Comment
Solubility ratio=1.04
Solubility ratio=1.083
Solubility ratio=1.059
Solubility ratio1.018Not Active
Solubility ratio=0.954
Solubility ratio=1.036
Solubility ratio=1.026
Solubility ratio=0.996
Solubility ratio=1.057
Solubility ratio=1.049
Solubility ratio=1.035
Solubility ratio=1.017
Solubility ratio=1.049
Solubility ratio=1.04
Solubility ratio=1.077
Solubility ratio=1.079
Solubility ratio=1.035
Solubility ratio=0.996
Solubility ratio=1.025
Solubility ratio=1.057
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL638278
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1984
Volume: 27
Issue: 8
First Page: 967
Last Page: 978
DOI: 10.1021/jm00374a006
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
Solubility=172200ug.mL-1Outside typical range
Solubility=183900ug.mL-1Outside typical range
Solubility=171400ug.mL-1Outside typical range
Solubility=175100ug.mL-1Outside typical range
Solubility=182400ug.mL-1Outside typical range
Solubility=173200ug.mL-1Outside typical range
Solubility=170700ug.mL-1Outside typical range
Solubility=177300ug.mL-1Outside typical range
Solubility=176200ug.mL-1Outside typical range
Solubility=166300ug.mL-1Outside typical range
Solubility=167000ug.mL-1Outside typical range
Solubility=170700ug.mL-1Outside typical range
Solubility=173600ug.mL-1Outside typical range
Solubility=166300ug.mL-1Outside typical range
Solubility=170700ug.mL-1Outside typical range
Solubility=172500ug.mL-1Outside typical range
Solubility=190500ug.mL-1Outside typical range
Solubility=175100ug.mL-1Outside typical range
Solubility=179500ug.mL-1Outside typical range
Solubility=167000ug.mL-1Outside typical range
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL638280
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1984
Volume: 27
Issue: 8
First Page: 967
Last Page: 978
DOI: 10.1021/jm00374a006
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
Solubility=249900ug.mL-1Outside typical range
Solubility=242400ug.mL-1Outside typical range
Solubility=249900ug.mL-1Outside typical range
Solubility=253600ug.mL-1Outside typical range
Solubility=248100ug.mL-1Outside typical range
Solubility=245000ug.mL-1Outside typical range
Solubility=230700ug.mL-1Outside typical range
Solubility=238700ug.mL-1Outside typical range
Solubility=246300ug.mL-1Outside typical range
Solubility=230700ug.mL-1Outside typical range
Solubility=234100ug.mL-1Outside typical range
Solubility=241500ug.mL-1Outside typical range
Solubility=238800ug.mL-1Outside typical range
Solubility=230700ug.mL-1Outside typical range
Solubility=230700ug.mL-1Outside typical range
Solubility=238700ug.mL-1Outside typical range
Solubility=242400ug.mL-1Outside typical range
Solubility=238700ug.mL-1Outside typical range
Solubility=242400ug.mL-1Outside typical range
Solubility=242900ug.mL-1Outside typical range
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL633104
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1984
Volume: 27
Issue: 8
First Page: 967
Last Page: 978
DOI: 10.1021/jm00374a006
Standard TypeStandard RelationStandard Value
Solubility ratio=1.073
Solubility ratio=1.162
Solubility ratio=1.118
Solubility ratio=1.064
Solubility ratio=0.932
Solubility ratio=1.048
Solubility ratio=1.069
Solubility ratio=1.012
Solubility ratio=1.134
Solubility ratio=1.093
Solubility ratio=1.086
Solubility ratio=1.036
Solubility ratio=1.083
Solubility ratio=1.046
Solubility ratio=1.043
Solubility ratio=1.13
Solubility ratio=1.027
Solubility ratio=1.004
Solubility ratio=1.057
Solubility ratio=1.123
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL633105
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1984
Volume: 27
Issue: 8
First Page: 967
Last Page: 978
DOI: 10.1021/jm00374a006
Standard TypeStandard RelationStandard Value
Solubility ratio=1.117
Solubility ratio=1.309
Solubility ratio=1.233
Solubility ratio=1.155
Solubility ratio=0.981
Solubility ratio=1.093
Solubility ratio=1.168
Solubility ratio=1.054
Solubility ratio=1.323
Solubility ratio=1.18
Solubility ratio=1.18
Solubility ratio=1.064
Solubility ratio=1.151
Solubility ratio=1.09
Solubility ratio=1.139
Solubility ratio=1.295
Solubility ratio=1.16
Solubility ratio=1.063
Solubility ratio=1.09
Solubility ratio=1.228