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90-07-3 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3301371
Protocol: N/A
Comment: Data Source: AstraZeneca DMPK/physicochemical
Standard TypeStandard RelationStandard ValueStandard Units
CL12.02uL.min-1.(10^6cells)-1
CL>150uL.min-1.(10^6cells)-1
CL13.18uL.min-1.(10^6cells)-1
CL>150uL.min-1.(10^6cells)-1
CL>150uL.min-1.(10^6cells)-1
CL>150uL.min-1.(10^6cells)-1
CL52uL.min-1.(10^6cells)-1
CL>150uL.min-1.(10^6cells)-1
CL<3uL.min-1.(10^6cells)-1
CL>150uL.min-1.(10^6cells)-1
CL144uL.min-1.(10^6cells)-1
CL11.75uL.min-1.(10^6cells)-1
CL<3uL.min-1.(10^6cells)-1
CL61uL.min-1.(10^6cells)-1
CL>150uL.min-1.(10^6cells)-1
CL24.55uL.min-1.(10^6cells)-1
CL14.24uL.min-1.(10^6cells)-1
CL13.18uL.min-1.(10^6cells)-1
CL<3uL.min-1.(10^6cells)-1
CL114uL.min-1.(10^6cells)-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3301370
Protocol: N/A
Comment: Data Source: AstraZeneca DMPK/physicochemical
Standard TypeStandard RelationStandard ValueStandard Units
CL8.33mL.min-1.g-1
CL4mL.min-1.g-1
CL13.49mL.min-1.g-1
CL48.98mL.min-1.g-1
CL5.75mL.min-1.g-1
CL6mL.min-1.g-1
CL<3mL.min-1.g-1
CL43.65mL.min-1.g-1
CL35mL.min-1.g-1
CL6.31mL.min-1.g-1
CL<3mL.min-1.g-1
CL15.14mL.min-1.g-1
CL<3mL.min-1.g-1
CL5.75mL.min-1.g-1
CL<3mL.min-1.g-1
CL82mL.min-1.g-1
CL29.51mL.min-1.g-1
CL6.46mL.min-1.g-1
CL116mL.min-1.g-1
CL8mL.min-1.g-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3301363
Protocol: N/A
Comment: Data Source: AstraZeneca DMPK/physicochemical
Standard TypeStandard Value
LogD7.41.56
LogD7.41.39
LogD7.4-0.78
LogD7.42.22
LogD7.43
LogD7.41.91
LogD7.4-0.84
LogD7.41.19
LogD7.4-1.08
LogD7.43.08
LogD7.43.65
LogD7.4-0.5
LogD7.42.43
LogD7.42.3
LogD7.43.65
LogD7.44.3
LogD7.43.26
LogD7.42.55
LogD7.41.69
LogD7.41.46
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3301365
Protocol: N/A
Comment: Data Source: AstraZeneca DMPK/physicochemical
Standard TypeStandard ValueStandard Units
PPB96%
PPB34.42%
PPB87.87%
PPB79.55%
PPB55.73%
PPB99.91%
PPB98.61%
PPB99.81%
PPB87.11%
PPB96.26%
PPB92.32%
PPB66.1%
PPB75.97%
PPB99.19%
PPB62.4%
PPB30.88%
PPB71.99%
PPB98.37%
PPB92.64%
PPB95.72%