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876-03-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:4-aminobutyrate aminotransferase, mitochondrial
External ID: CHEMBL939956
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2008
Volume: 18
Issue: 10
First Page: 3122
Last Page: 3125
DOI: 10.1016/j.bmcl.2007.10.060

Target ChEMBL ID: CHEMBL2044
ChEMBL Target Name: Gamma-amino-N-butyrate transaminase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
Relative stimulatory activity=0%
Relative stimulatory activity=0%
Relative stimulatory activity=0%
Relative stimulatory activity=0.78%
Relative stimulatory activity=5.65%
Relative stimulatory activity=0%
Relative stimulatory activity=3.42%