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867331-64-4 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:HepG2
External ID: CHEMBL5303715
Protocol: N/A
Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Target ChEMBL ID: CHEMBL395
ChEMBL Target Name: HepG2
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Data Source: EU-OPENSCREEN
PubChem Standard ValueStandard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
2.8IC50 relative=2800nMActive
8.5IC50 relative=8500nMActive
8.2IC50 relative=8200nMActive
8.7IC50 relative=8700nMActive
15IC50 relative=15000nMInactive
1.1IC50 relative=1100nMActive
8.3IC50 relative=8300nMActive
7.8IC50 relative=7800nMActive
5.3IC50 relative=5300nMActive
4.5IC50 relative=4500nMActive
2.5IC50 relative=2500nMActive
12.5IC50 relative=12500nMInactive
1IC50 relative=1000nMActive
0.7IC50 relative=700nMActive
3.6IC50 relative=3600nMActive
2.7IC50 relative=2700nMActive
13.1IC50 relative=13100nMActive
1.9IC50 relative=1900nMActive
11.8IC50 relative=11800nMInactive
50IC50 relative=50000nMInactive