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83807-07-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Estrogen receptor beta
External ID: CHEMBL781841
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1983
Volume: 26
Issue: 8
First Page: 1131
Last Page: 1137
DOI: 10.1021/jm00362a009

Target ChEMBL ID: CHEMBL2094114
ChEMBL Target Name: Estrogen receptor
ChEMBL Target Type: PROTEIN FAMILY - Target is a group of closely related proteins
Relationship Type: D - Direct protein target assigned
Confidence: Multiple direct protein targets may be assigned
Standard TypeStandard Relation
Activity=
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL742683
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1983
Volume: 26
Issue: 8
First Page: 1131
Last Page: 1137
DOI: 10.1021/jm00362a009

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeActivity CommentData Validity Comment
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
ActivityNo dataPotential missing data
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Estrogen receptor beta
External ID: CHEMBL674366
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1983
Volume: 26
Issue: 8
First Page: 1131
Last Page: 1137
DOI: 10.1021/jm00362a009

Target ChEMBL ID: CHEMBL2094114
ChEMBL Target Name: Estrogen receptor
ChEMBL Target Type: PROTEIN FAMILY - Target is a group of closely related proteins
Relationship Type: H - Homologous protein target assigned
Confidence: Multiple homologous protein targets may be assigned
Standard TypeStandard RelationStandard Value
RBA=5.9
RBA=0.54
RBA=0.02
RBA=0.02
RBA=0.22
RBA=6.1
RBA=0.12
RBA=0.65
RBA=0.36
RBA=50
RBA=0.12
RBA=0.1
RBA=0.07
RBA=15
RBA=5.2
RBA=9.2
RBA=5
RBA=0.21
RBA=52
RBA=9.1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Rattus norvegicus
External ID: CHEMBL777446
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1983
Volume: 26
Issue: 8
First Page: 1131
Last Page: 1137
DOI: 10.1021/jm00362a009

Target ChEMBL ID: CHEMBL376
ChEMBL Target Name: Rattus norvegicus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard UnitsActivity Comment
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
DOSEmg.kg-1Not Determined
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Rattus norvegicus
External ID: CHEMBL789221
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1983
Volume: 26
Issue: 8
First Page: 1131
Last Page: 1137
DOI: 10.1021/jm00362a009

Target ChEMBL ID: CHEMBL376
ChEMBL Target Name: Rattus norvegicus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MFED>25mg kg-1
MFED=25mg kg-1
MFED=10mg kg-1
MFED>25mg kg-1
MFED=10mg kg-1
MFED=5mg kg-1
MFED=25mg kg-1
MFED=5mg kg-1
MFED>25mg kg-1
MFED=0.5mg kg-1
MFED=5mg kg-1
MFED=0.5mg kg-1
MFED=0.5mg kg-1
MFED=25mg kg-1
MFED=5mg kg-1