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80353-09-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Amine oxidase [flavin-containing] B
External ID: CHEMBL715309
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1993
Volume: 36
Issue: 9
First Page: 1278
Last Page: 1283
DOI: 10.1021/jm00061a020

Target ChEMBL ID: CHEMBL2756
ChEMBL Target Name: Monoamine oxidase B
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
TN=283uM min-1
TN=61uM min-1
TN=204uM min-1
TN=337uM min-1
TN=165uM min-1
TN=4.17uM min-1
TN=12uM min-1
TN=193uM min-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Amine oxidase [flavin-containing] B
External ID: CHEMBL850386
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1993
Volume: 36
Issue: 9
First Page: 1278
Last Page: 1283
DOI: 10.1021/jm00061a020

Target ChEMBL ID: CHEMBL2756
ChEMBL Target Name: Monoamine oxidase B
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard Value
Ratio=963
Ratio=1130
Ratio=523
Ratio=3270
Ratio=71
Ratio=1250
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Amine oxidase [flavin-containing] B
External ID: CHEMBL732525
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 19
First Page: 3694
Last Page: 3700
DOI: 10.1021/jm9603882

Target ChEMBL ID: CHEMBL2756
ChEMBL Target Name: Monoamine oxidase B
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard Value
Ratio=1130
Ratio=55
Ratio=3580
Ratio=382
Ratio=92
Ratio=688
Ratio=4
Ratio=433
Ratio=16
Ratio=974
Ratio=54
Ratio=790
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Amine oxidase [flavin-containing] B
External ID: CHEMBL734660
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1993
Volume: 36
Issue: 20
First Page: 2929
Last Page: 2937
DOI: 10.1021/jm00072a012

Target ChEMBL ID: CHEMBL2095205
ChEMBL Target Name: Monoamine oxidase
ChEMBL Target Type: PROTEIN FAMILY - Target is a group of closely related proteins
Relationship Type: H - Homologous protein target assigned
Confidence: Multiple homologous protein targets may be assigned
Standard TypeStandard RelationStandard Value
Relative activity=3
Relative activity=2
Relative activity=3
Relative activity=2
Relative activity=3
Relative activity=3
Relative activity=3
Relative activity=3
Relative activity=2
Relative activity=3
Relative activity=2
Relative activity=3
Relative activity=2
Relative activity=2
Relative activity=3
Relative activity=1
Relative activity=2
Relative activity=2
Relative activity=2
Relative activity=3
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Amine oxidase [flavin-containing] A
External ID: CHEMBL715301
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1993
Volume: 36
Issue: 9
First Page: 1278
Last Page: 1283
DOI: 10.1021/jm00061a020

Target ChEMBL ID: CHEMBL1951
ChEMBL Target Name: Monoamine oxidase A
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
TN=10uM min-1
TN=137uM min-1
TN=20uM min-1
TN=8.4uM min-1
TN=146uM min-1
TN=8.14uM min-1
TN=5.21uM min-1
TN=9.2uM min-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Amine oxidase [flavin-containing] B
External ID: CHEMBL850385
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1993
Volume: 36
Issue: 9
First Page: 1278
Last Page: 1283
DOI: 10.1021/jm00061a020

Target ChEMBL ID: CHEMBL2756
ChEMBL Target Name: Monoamine oxidase B
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard Value
Ratio=13
Ratio=1120
Ratio=143
Ratio=175
Ratio=860
Ratio=80
Ratio=160
Ratio=28
Ratio=139