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74299-48-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Estrogen receptor
External ID: CHEMBL1941569
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2012
Volume: 22
Issue: 1
First Page: 154
Last Page: 163
DOI: 10.1016/j.bmcl.2011.11.041

Target ChEMBL ID: CHEMBL206
ChEMBL Target Name: Estrogen receptor alpha
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
Activity=48.44%
Activity=70%
Activity=141.67%
Activity=58.49%
Activity=64.78%
Activity=52.2%
Activity=62.16%
Activity=100%
Activity=36.36%
Activity=24.73%
Activity=12%
Activity=45.15%
Activity=60.45%
Activity=14.91%
Activity=92.19%
Activity=79.69%
Activity=22.91%
Activity=113.51%
Activity=34.7%
Activity=40.3%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Estrogen receptor
External ID: CHEMBL1941568
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2012
Volume: 22
Issue: 1
First Page: 154
Last Page: 163
DOI: 10.1016/j.bmcl.2011.11.041

Target ChEMBL ID: CHEMBL206
ChEMBL Target Name: Estrogen receptor alpha
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
Activity=71.77%
Activity=76.81%
Activity=234.78%
Activity=51.41%
Activity=46.89%
Activity=71.19%
Activity=2.78%
Activity=91.35%
Activity=37.3%
Activity=20%
Activity=25.95%
Activity=38.56%
Activity=75.42%
Activity=55.14%
Activity=63.71%
Activity=1.61%
Activity=25.95%
Activity=98.61%
Activity=34.75%
Activity=47.03%