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72049-24-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Acetylcholinesterase
External ID: CHEMBL2341264
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem.
Year: 2013
Volume: 21
Issue: 5
First Page: 1064
Last Page: 1073
DOI: 10.1016/j.bmc.2013.01.015

Target ChEMBL ID: CHEMBL3199
ChEMBL Target Name: Acetylcholinesterase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=32.87%
Inhibition<10%
Inhibition=53.16%
Inhibition=69.86%
Inhibition=43.03%
Inhibition=27.39%
Inhibition=101.51%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL661570
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 7
First Page: 817
Last Page: 822
DOI: 10.1016/S0960-894X(97)00102-9
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
Inhibition=3%
Inhibition=180%Outside typical range
Inhibition=81.8%
Inhibition=24.9%
Inhibition=4.8%
Inhibition=-1.9%
Inhibition=14.8%
Inhibition=18.5%
Inhibition=12.1%