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7161-63-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:BindingDB 靶标:N/A
External ID: BindingDB_8127_1
Protocol: N/A
Comment: Compounds with any of Ki, IC50, Kd, or EC50 activity value <= 10uM are labeled as "Active".
If multiple measurements are available for a given compound, it is labeled as "Active" if any of the measurements meet the criterion. Activity values are checked in the order of Ki, IC50, Kd, and EC50. The first entry that meets the above activity threshold is used to determine "Standard Type", "Standard Relation", and "PubChem Standard Value". Otherwise, the first non-empty entry will be used to set those values.
Standard TypePubChem Standard ValueIC50Target Accession(s)LigandTarget
IC5025.7425740P00533BDBM49214Epidermal growth factor receptor [645-1186]
IC505050000P00533BDBM234300Epidermal growth factor receptor [645-1186]
IC5024.8324830P00533BDBM234301Epidermal growth factor receptor [645-1186]
IC5014.1814180P00533BDBM234302Epidermal growth factor receptor [645-1186]
IC5021.9221920P00533BDBM234303Epidermal growth factor receptor [645-1186]
IC505050000P00533BDBM234304Epidermal growth factor receptor [645-1186]
IC5041.7641760P00533BDBM234305Epidermal growth factor receptor [645-1186]
IC505050000P00533BDBM234306Epidermal growth factor receptor [645-1186]
IC505050000P00533BDBM234307Epidermal growth factor receptor [645-1186]
IC5045.2945290P00533BDBM234308Epidermal growth factor receptor [645-1186]
IC5039.9839980P00533BDBM234309Epidermal growth factor receptor [645-1186]
IC5029.6229620P00533BDBM234310Epidermal growth factor receptor [645-1186]
IC505050000P00533BDBM234311Epidermal growth factor receptor [645-1186]
IC5022.1922190P00533BDBM234312Epidermal growth factor receptor [645-1186]
IC5040.1740170P00533BDBM234313Epidermal growth factor receptor [645-1186]
IC505050000P00533BDBM234314Epidermal growth factor receptor [645-1186]
IC505050000P00533BDBM234315Epidermal growth factor receptor [645-1186]
IC5031.0931090P00533BDBM234316Epidermal growth factor receptor [645-1186]
IC5034.6734670P00533BDBM234317Epidermal growth factor receptor [645-1186]
IC505050000P00533BDBM234318Epidermal growth factor receptor [645-1186]