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7069-41-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:HTH-type transcriptional regulator LuxR
External ID: CHEMBL5265248
Protocol: N/A
Comment: Journal: Eur J Med Chem
Year: 2020
Volume: 207
First Page: 112741
Last Page: 112741
DOI: 10.1016/j.ejmech.2020.112741

Target ChEMBL ID: CHEMBL5291573
ChEMBL Target Name: HTH-type transcriptional regulator LuxR
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=62%
Inhibition=65%
Inhibition=78%
Inhibition=14%
Inhibition=100%
Inhibition=58%
Inhibition=34%
Inhibition=55%
Inhibition=71%
Inhibition=100%
Inhibition=90%
Inhibition=94%
Inhibition=17%
Inhibition=13%
Inhibition=56%
Inhibition=35%
Inhibition=87%
Inhibition=59%
Inhibition=80%
Inhibition=73%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Bursaphelenchus xylophilus
External ID: CHEMBL3048285
Protocol: N/A
Comment: Journal: J Agric Food Chem
Year: 2010
Volume: 58
Issue: 3
First Page: 1823
Last Page: 1827
DOI: 10.1021/jf902575f

Target ChEMBL ID: CHEMBL613331
ChEMBL Target Name: Bursaphelenchus xylophilus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
mortality=12.6%
mortality=31.3%
mortality=29.8%
mortality=4.4%
mortality=13.6%
mortality=6%
mortality=4.2%
mortality=3.1%
mortality=100%
mortality=100%
mortality=100%
mortality=100%
mortality=4.4%
mortality=4%
mortality=1.6%
mortality=4.4%
mortality=98.5%
mortality=100%
mortality=3.8%
mortality=100%