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6975-73-1 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3755087
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 3
First Page: 978
Last Page: 985
DOI: 10.1016/j.bmcl.2015.12.049
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
IC50>100ug.mL-1Outside typical range
IC50=60ug.mL-1Outside typical range
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL3755086
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 3
First Page: 978
Last Page: 985
DOI: 10.1016/j.bmcl.2015.12.049

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
MIC=20ug.mL-1
MIC>20ug.mL-1
MIC>20ug.mL-1
MIC>20ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL3755085
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 3
First Page: 978
Last Page: 985
DOI: 10.1016/j.bmcl.2015.12.049

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
MIC=0.06ug.mL-1
MIC=5ug.mL-1
MIC=5.2ug.mL-1
MIC>10ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3755088
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 3
First Page: 978
Last Page: 985
DOI: 10.1016/j.bmcl.2015.12.049
Standard TypeStandard RelationStandard Value
Selectivity Index>1666
Selectivity Index=11.5