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69159-51-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL3231029
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1979
Volume: 22
Issue: 2
First Page: 183
Last Page: 191
DOI: 10.1021/jm00188a012

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
ED50=1.6mg.kg-1
ED50=1.3mg.kg-1
ED50=24mg.kg-1
ED50=21.8mg.kg-1
ED50>25mg.kg-1
ED50>12.5mg.kg-1
ED50=3.5mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50=5mg.kg-1
ED50=2.9mg.kg-1
ED50=10mg.kg-1
ED50=6.5mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50=12mg.kg-1
ED50=7mg.kg-1
ED50=17mg.kg-1
ED50>25mg.kg-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL3231032
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1979
Volume: 22
Issue: 2
First Page: 183
Last Page: 191
DOI: 10.1021/jm00188a012

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
ED50=19.4mg.kg-1
ED50=8mg.kg-1
ED50>50mg.kg-1
ED50>50mg.kg-1
ED50=28mg.kg-1
ED50>12.5mg.kg-1
ED50=9.6mg.kg-1
ED50=45mg.kg-1
ED50>50mg.kg-1
ED50>50mg.kg-1
ED50=17mg.kg-1
ED50=13.4mg.kg-1
ED50=16.7mg.kg-1
ED50=23.3mg.kg-1
ED50=28.7mg.kg-1
ED50>50mg.kg-1
ED50>50mg.kg-1
ED50=21.5mg.kg-1
ED50=46.9mg.kg-1
ED50=31mg.kg-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL3231031
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1979
Volume: 22
Issue: 2
First Page: 183
Last Page: 191
DOI: 10.1021/jm00188a012

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
ED50=12.3mg.kg-1
ED50=6.6mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50=12.5mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50=12mg.kg-1
ED50=7.3mg.kg-1
ED50=12.5mg.kg-1
ED50=8.5mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
ED50=12.5mg.kg-1
ED50>25mg.kg-1
ED50>25mg.kg-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL3231033
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1979
Volume: 22
Issue: 2
First Page: 183
Last Page: 191
DOI: 10.1021/jm00188a012

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
LD50=200mg.kg-1
LD50=100mg.kg-1
LD50=50mg.kg-1
LD50=400mg.kg-1
LD50=400mg.kg-1
LD50=400mg.kg-1
LD50=200mg.kg-1
LD50=200mg.kg-1
LD50=400mg.kg-1
LD50=200mg.kg-1
LD50=200mg.kg-1
LD50=400mg.kg-1
LD50=200mg.kg-1
LD50=200mg.kg-1
LD50=400mg.kg-1
LD50=400mg.kg-1
LD50=800mg.kg-1
LD50=400mg.kg-1
LD50>800mg.kg-1
LD50=400mg.kg-1