HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：High affinity choline transporter 1

External ID: CHEMBL1211032

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg Med Chem Lett
Year: 2010
Volume: 20
Issue: 16
First Page: 4870
Last Page: 4877
DOI: 10.1016/j.bmcl.2010.06.090

Target ChEMBL ID: CHEMBL3013
ChEMBL Target Name: Choline transporter
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units	Data Validity Comment
340.017	Ki	=	340016.51	nM	Outside typical range
0.68077	Ki	=	680.77	nM
32.0627	Ki	=	32062.69	nM
35075.2	Ki	=	3.50751874E7	nM	Outside typical range
55.7186	Ki	=	55718.57	nM
3801.89	Ki	=	3801893.96	nM	Outside typical range
150003	Ki	=	1.5000301905E8	nM	Outside typical range
9418.9	Ki	=	9418895.97	nM	Outside typical range
820.352	Ki	=	820351.54	nM	Outside typical range
1051.96	Ki	=	1051961.87	nM	Outside typical range
75.1623	Ki	=	75162.29	nM
2.20293	Ki	=	2202.93	nM
310.456	Ki	=	310455.96	nM	Outside typical range
290.402	Ki	=	290402.27	nM	Outside typical range
190.108	Ki	=	190107.83	nM	Outside typical range
270.023	Ki	=	270022.53	nM	Outside typical range
340.017	Ki	=	340016.51	nM	Outside typical range
2.00032	Ki	=	2000.32	nM
40.0867	Ki	=	40086.67	nM
210.378	Ki	=	210377.84	nM	Outside typical range

6701-82-2 靶点实验数据