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64357-53-5 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Leishmania amazonensis
External ID: CHEMBL2416389
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem.
Year: 2013
Volume: 21
Issue: 11
First Page: 3114
Last Page: 3119
DOI: 10.1016/j.bmc.2013.03.045

Target ChEMBL ID: CHEMBL612877
ChEMBL Target Name: Leishmania amazonensis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
IC50=0.44ug.mL-1
IC50=4.7ug.mL-1
IC50=40.92ug.mL-1
IC50=29ug.mL-1
IC50=121.36ug.mL-1Outside typical range
IC50=5.05ug.mL-1
IC50=4.9ug.mL-1
IC50=8.56ug.mL-1
IC50=9.8ug.mL-1
IC50=7.82ug.mL-1
IC50=21.3ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL2416388
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem.
Year: 2013
Volume: 21
Issue: 11
First Page: 3114
Last Page: 3119
DOI: 10.1016/j.bmc.2013.03.045
Standard TypeStandard RelationStandard ValueStandard Units
CC50=3.82ug.mL-1
CC50=25ug.mL-1
CC50>160ug.mL-1
CC50>160ug.mL-1
CC50>160ug.mL-1
CC50=28ug.mL-1
CC50=24.6ug.mL-1
CC50=28.9ug.mL-1
CC50=40.6ug.mL-1
CC50=87.1ug.mL-1
CC50=116.2ug.mL-1