HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Bifunctional epoxide hydrolase 2

External ID: CHEMBL999421

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg Med Chem Lett
Year: 2009
Volume: 19
Issue: 8
First Page: 2354
Last Page: 2359
DOI: 10.1016/j.bmcl.2008.09.066

Target ChEMBL ID: CHEMBL2409
ChEMBL Target Name: Epoxide hydratase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units	Activity Comment
0.0336	IC50	=	33.6	nM
	IC50				Not Determined
	IC50				Not Determined

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Bifunctional epoxide hydrolase 2

External ID: CHEMBL999422

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2009
Volume: 19
Issue: 8
First Page: 2354
Last Page: 2359
DOI: 10.1016/j.bmcl.2008.09.066

Target ChEMBL ID: CHEMBL2409
ChEMBL Target Name: Epoxide hydratase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	92	%
Inhibition	=	90	%
Inhibition	=	75	%

640259-75-2 靶点实验数据