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598-75-4 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Tetrahymena pyriformis
External ID: CHEMBL3057542
Protocol: N/A
Comment: Journal: Med Chem Res
Year: 2009
Volume: 18
Issue: 9
First Page: 770
Last Page: 781
DOI: 10.1007/s00044-009-9166-z

Target ChEMBL ID: CHEMBL612891
ChEMBL Target Name: Tetrahymena pyriformis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
PubChem Standard ValueStandard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
785236GI50=7.8523563461E8nMOutside typical range
17930.8GI50=1.793081377E7nMOutside typical range
2159.73GI50=2159732.68nM
10204.7GI50=1.020469432E7nMOutside typical range
16177.1GI50=1.617707504E7nMOutside typical range
13125GI50=1.312502079E7nMOutside typical range
183316GI50=1.8331584287E8nMOutside typical range
28707.8GI50=2.870780582E7nMOutside typical range
57055.8GI50=5.705582639E7nMOutside typical range
69246.8GI50=6.924684643E7nMOutside typical range
67158.3GI50=6.715834729E7nMOutside typical range
29221.3GI50=2.922133142E7nMOutside typical range
442792GI50=4.4279223878E8nMOutside typical range
111481GI50=1.1148078034E8nMOutside typical range
92066.2GI50=9.206615375E7nMOutside typical range
100949GI50=1.0094853019E8nMOutside typical range
134834GI50=1.3483418052E8nMOutside typical range
68833.5GI50=6.883352333E7nMOutside typical range
267855GI50=2.6785514945E8nMOutside typical range
118468GI50=1.1846771176E8nMOutside typical range
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL938588
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem.
Year: 2009
Volume: 17
Issue: 2
First Page: 896
Last Page: 904
DOI: 10.1016/j.bmc.2008.11.040
Standard TypeStandard RelationStandard Value
log Ks=2.33
log Ks=2.76
log Ks=1.76
log Ks=1.78
log Ks=1.97
log Ks=2.52
log Ks=3.28
log Ks=2.71
log Ks=3.22
log Ks=1.78
log Ks=3.01
log Ks=3.07
log Ks=3.08
log Ks=1.98
log Ks=2.32
log Ks=2.2
log Ks=2.67
log Ks=2.69
log Ks=1.73
log Ks=1.97