HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：HT-29

External ID: CHEMBL905029

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg. Med. Chem.
Year: 2007
Volume: 15
Issue: 13
First Page: 4456
Last Page: 4469
DOI: 10.1016/j.bmc.2007.04.028

Target ChEMBL ID: CHEMBL384
ChEMBL Target Name: HT-29
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units	Activity Comment
4.7	GI50	=	4700	nM
1.9	GI50	=	1900	nM
2.3	GI50	=	2300	nM
15	GI50	=	15000	nM
	Activity				Not Evaluated
16	GI50	=	16000	nM
8.5	GI50	=	8500	nM
	Activity				Not Evaluated
39	GI50	=	39000	nM
	Activity				Not Evaluated
78	GI50	=	78000	nM
95	GI50	=	95000	nM
2.3	GI50	=	2300	nM
33	GI50	=	33000	nM
13	GI50	=	13000	nM
9	GI50	=	9000	nM
15	GI50	=	15000	nM
44	GI50	=	44000	nM
2.7	GI50	=	2700	nM
4.9	GI50	=	4900	nM

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：M21

External ID: CHEMBL904042

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg. Med. Chem.
Year: 2007
Volume: 15
Issue: 13
First Page: 4456
Last Page: 4469
DOI: 10.1016/j.bmc.2007.04.028

Target ChEMBL ID: CHEMBL614117
ChEMBL Target Name: M21
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units	Activity Comment
8.9	GI50	=	8900	nM
3.9	GI50	=	3900	nM
4.3	GI50	=	4300	nM
27	GI50	=	27000	nM
	Activity				Not Evaluated
33	GI50	=	33000	nM
16	GI50	=	16000	nM
	Activity				Not Evaluated
81	GI50	=	81000	nM
	Activity				Not Evaluated
	Activity				Not Evaluated
	Activity				Not Evaluated
5.1	GI50	=	5100	nM
61	GI50	=	61000	nM
22	GI50	=	22000	nM
17	GI50	=	17000	nM
26	GI50	=	26000	nM
73	GI50	=	73000	nM
5.1	GI50	=	5100	nM
8.1	GI50	=	8100	nM

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：MCF7

External ID: CHEMBL904043

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg. Med. Chem.
Year: 2007
Volume: 15
Issue: 13
First Page: 4456
Last Page: 4469
DOI: 10.1016/j.bmc.2007.04.028

Target ChEMBL ID: CHEMBL387
ChEMBL Target Name: MCF7
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units	Activity Comment
17	GI50	=	17000	nM
6	GI50	=	6000	nM
6.2	GI50	=	6200	nM
23	GI50	=	23000	nM
	Activity				Not Evaluated
44	GI50	=	44000	nM
31	GI50	=	31000	nM
	Activity				Not Evaluated
	Activity				Not Evaluated
	Activity				Not Evaluated
	Activity				Not Evaluated
	Activity				Not Evaluated
14.2	GI50	=	14200	nM
52	GI50	=	52000	nM
27	GI50	=	27000	nM
15	GI50	=	15000	nM
23	GI50	=	23000	nM
72	GI50	=	72000	nM
5.7	GI50	=	5700	nM
9.1	GI50	=	9100	nM

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：M21

External ID: CHEMBL905030

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem.
Year: 2007
Volume: 15
Issue: 13
First Page: 4456
Last Page: 4469
DOI: 10.1016/j.bmc.2007.04.028

Target ChEMBL ID: CHEMBL614117
ChEMBL Target Name: M21
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Activity Comment
Activity	Not Active
Activity	Not Active
Activity	Not Active
Activity	Not Active
Activity	Not Active
Activity	Not Active
Activity	Not Active
Activity	Not Active

5544-33-2 靶点实验数据