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5259-86-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3280532
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1977
Volume: 20
Issue: 2
First Page: 233
Last Page: 236
DOI: 10.1021/jm00212a009
Standard TypeStandard RelationStandard ValueActivity Comment
Inhibition_index=260
Inhibition_indexNot Determined
Inhibition_index=600
Inhibition_index=1000
Inhibition_index=600
Inhibition_indexNot Determined
Inhibition_index=800
Inhibition_index=53
Inhibition_index=120
Inhibition_index=800
Inhibition_index=450
Inhibition_indexNot Determined
Inhibition_index=400
Inhibition_index=210
Inhibition_index=180
Inhibition_index=105
Inhibition_index=76
Inhibition_index=250
Inhibition_index=700
Inhibition_index=600
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3284061
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1977
Volume: 20
Issue: 11
First Page: 1420
Last Page: 1435
DOI: 10.1021/jm00221a013
Standard TypeStandard RelationStandard Value
log(1/Km)=2.12
log(1/Km)=2.08
log(1/Km)=1.19
log(1/Km)=1.27
log(1/Km)=1.51
log(1/Km)=1.62
log(1/Km)=1.71
log(1/Km)=1.75
log(1/Km)=2.1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3284068
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1977
Volume: 20
Issue: 11
First Page: 1420
Last Page: 1435
DOI: 10.1021/jm00221a013
Standard TypeStandard RelationStandard Value
logKcat=-1.39
logKcat=-1.42
logKcat=-0.88
logKcat=-1.07
logKcat=-1.89
logKcat=-1.6
logKcat=-0.01
logKcat=-0.8
logKcat=-2.22