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520-68-3 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:CHO
External ID: CHEMBL3054995
Protocol: N/A
Comment: Journal: Biochem Syst Ecol
Year: 2008
Volume: 36
Issue: 3
First Page: 153
Last Page: 166
DOI: 10.1016/jbse.2007.08.015

Target ChEMBL ID: CHEMBL613853
ChEMBL Target Name: CHO
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity CommentData Validity Comment
EC50>100ug.mL-1Outside typical range
EC50>100ug.mL-1Outside typical range
EC50Not Determined
EC50>100ug.mL-1Outside typical range
EC50>100ug.mL-1Outside typical range
EC50>100ug.mL-1Outside typical range
EC50>100ug.mL-1Outside typical range
EC50Not Determined
EC50Not Determined
EC50=13.2ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3054470
Protocol: N/A
Comment: Journal: Biochem Syst Ecol
Year: 2008
Volume: 36
Issue: 3
First Page: 153
Last Page: 166
DOI: 10.1016/jbse.2007.08.015
Standard TypeStandard RelationStandard ValueStandard UnitsActivity CommentData Validity Comment
EC50>100ug.mL-1Outside typical range
EC50>100ug.mL-1Outside typical range
EC50Not Determined
EC50>100ug.mL-1Outside typical range
EC50>100ug.mL-1Outside typical range
EC50>100ug.mL-1Outside typical range
EC50>100ug.mL-1Outside typical range
EC50Not Determined
EC50Not Determined
EC50>100ug.mL-1Outside typical range
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Spodoptera littoralis
External ID: CHEMBL3054471
Protocol: N/A
Comment: Journal: Biochem Syst Ecol
Year: 2008
Volume: 36
Issue: 3
First Page: 153
Last Page: 166
DOI: 10.1016/jbse.2007.08.015

Target ChEMBL ID: CHEMBL612897
ChEMBL Target Name: Spodoptera littoralis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity=84%
Activity=47%
Activity=116%
Activity=89%
Activity=102%
Activity=90%
Activity=87%
Activity=90%
Activity=118%
Activity=102%
Activity=90%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Spodoptera littoralis
External ID: CHEMBL3054472
Protocol: N/A
Comment: Journal: Biochem Syst Ecol
Year: 2008
Volume: 36
Issue: 3
First Page: 153
Last Page: 166
DOI: 10.1016/jbse.2007.08.015

Target ChEMBL ID: CHEMBL612897
ChEMBL Target Name: Spodoptera littoralis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity=84%
Activity=98%
Activity=105%
Activity=88%
Activity=92%
Activity=88%
Activity=82%
Activity=97%
Activity=165%
Activity=113%
Activity=98%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Rhopalosiphum padi
External ID: CHEMBL3054473
Protocol: N/A
Comment: Journal: Biochem Syst Ecol
Year: 2008
Volume: 36
Issue: 3
First Page: 153
Last Page: 166
DOI: 10.1016/jbse.2007.08.015

Target ChEMBL ID: CHEMBL2366656
ChEMBL Target Name: Rhopalosiphum padi
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
Activity=40%
Activity=37%
Activity=53%
Activity=43%
Activity=40%
Activity=46%
Activity=42%
Activity=42%
Activity=36%
Activity=43%
ActivityNot Determined
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Myzus persicae
External ID: CHEMBL3054474
Protocol: N/A
Comment: Journal: Biochem Syst Ecol
Year: 2008
Volume: 36
Issue: 3
First Page: 153
Last Page: 166
DOI: 10.1016/jbse.2007.08.015

Target ChEMBL ID: CHEMBL612683
ChEMBL Target Name: Myzus persicae
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
Activity=40%
Activity=49%
Activity=35%
Activity=57%
Activity=30%
Activity=44%
Activity=50%
Activity=35%
Activity=40%
Activity=40%
ActivityNot Determined
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Leptinotarsa decemlineata
External ID: CHEMBL3054475
Protocol: N/A
Comment: Journal: Biochem Syst Ecol
Year: 2008
Volume: 36
Issue: 3
First Page: 153
Last Page: 166
DOI: 10.1016/jbse.2007.08.015

Target ChEMBL ID: CHEMBL613217
ChEMBL Target Name: Leptinotarsa decemlineata
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
EC50=1.3microg/cm2
EC50>50microg/cm2
EC50>50microg/cm2
EC50=3.4microg/cm2
EC50Not Determined
EC50>50microg/cm2
EC50=1.7microg/cm2
EC50=4.8microg/cm2
EC50=1.4microg/cm2
EC50>50microg/cm2
EC50>50microg/cm2
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Spodoptera littoralis
External ID: CHEMBL3054476
Protocol: N/A
Comment: Journal: Biochem Syst Ecol
Year: 2008
Volume: 36
Issue: 3
First Page: 153
Last Page: 166
DOI: 10.1016/jbse.2007.08.015

Target ChEMBL ID: CHEMBL612897
ChEMBL Target Name: Spodoptera littoralis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
EC50>50microg/cm2
EC50>50microg/cm2
EC50>50microg/cm2
EC50>100microg/cm2
EC50Not Determined
EC50>50microg/cm2
EC50=50microg/cm2
EC50=0.2microg/cm2
EC50>50microg/cm2
EC50>50microg/cm2
EC50>50microg/cm2