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483-90-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Acetylcholinesterase
External ID: CHEMBL3068057
Protocol: N/A
Comment: Journal: Med Chem Res
Year: 2012
Volume: 21
Issue: 6
First Page: 722
Last Page: 725
DOI: 10.1007/s00044-011-9581-9

Target ChEMBL ID: CHEMBL220
ChEMBL Target Name: Acetylcholinesterase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard UnitsActivity CommentData Validity Comment
IC50=0.013ug.mL-1
IC50=8.6ug.mL-1
IC50Not Active
IC50Not Active
IC50>100ug.mL-1Outside typical range
IC50>100ug.mL-1Outside typical range
IC50Not Active
IC50Not Active
IC50Not Active
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Acetylcholinesterase
External ID: CHEMBL3068058
Protocol: N/A
Comment: Journal: Med Chem Res
Year: 2012
Volume: 21
Issue: 6
First Page: 722
Last Page: 725
DOI: 10.1007/s00044-011-9581-9

Target ChEMBL ID: CHEMBL220
ChEMBL Target Name: Acetylcholinesterase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=91.3%
Inhibition=12.6%
Inhibition=24.3%
Inhibition=51.9%
Inhibition=49.7%
Inhibition=9.9%
Inhibition=33.9%
Inhibition=34.4%