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4697-36-3 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Proteus mirabilis
External ID: CHEMBL768999
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1980
Volume: 23
Issue: 4
First Page: 405
Last Page: 412
DOI: 10.1021/jm00178a011

Target ChEMBL ID: CHEMBL614444
ChEMBL Target Name: Proteus mirabilis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=12.5ug.mL-1
MIC=0.4ug.mL-1
MIC=0.8ug.mL-1
MIC=12.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267883
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=2ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=0.25ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=1ug.mL-1
MIC=1ug.mL-1
MIC=156ug.mL-1
MIC=0.031ug.mL-1
MIC=1ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267884
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=2ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=0.25ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=1ug.mL-1
MIC=156ug.mL-1
MIC=0.031ug.mL-1
MIC=1ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267893
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=2ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=4ug.mL-1
MIC=1ug.mL-1
MIC=2500ug.mL-1
MIC=0.031ug.mL-1
MIC=1ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267885
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=4ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=1ug.mL-1
MIC=5000ug.mL-1
MIC=0.031ug.mL-1
MIC=1ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267886
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=4ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=1ug.mL-1
MIC=5000ug.mL-1
MIC=0.031ug.mL-1
MIC=1ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267887
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
MIC=8ug.mL-1
MIC=2ug.mL-1
MIC=0.063ug.mL-1
MIC=2ug.mL-1
MIC=0.13ug.mL-1
MIC=2ug.mL-1
MIC=4ug.mL-1
MIC=4ug.mL-1
MIC=10000ug.mL-1Outside typical range
MIC=0.063ug.mL-1
MIC=2ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267888
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=4ug.mL-1
MIC=1ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=1ug.mL-1
MIC=5000ug.mL-1
MIC=0.031ug.mL-1
MIC=2ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267889
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=4ug.mL-1
MIC=1ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=1ug.mL-1
MIC=5000ug.mL-1
MIC=0.031ug.mL-1
MIC=2ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267890
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
MIC=8ug.mL-1
MIC=4ug.mL-1
MIC=0.25ug.mL-1
MIC=4ug.mL-1
MIC=0.13ug.mL-1
MIC=4ug.mL-1
MIC=8ug.mL-1
MIC=4ug.mL-1
MIC=10000ug.mL-1Outside typical range
MIC=0.13ug.mL-1
MIC=8ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267891
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=2ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=1ug.mL-1
MIC=2500ug.mL-1
MIC=0.031ug.mL-1
MIC=1ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1267892
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2010
Volume: 54
Issue: 5
First Page: 2239
Last Page: 2243
DOI: 10.1128/aac.01677-09

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=2ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=0.5ug.mL-1
MIC=0.063ug.mL-1
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=1ug.mL-1
MIC=2500ug.mL-1
MIC=0.031ug.mL-1
MIC=1ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675395
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>125ug.mL-1
MIC>125ug.mL-1
MIC=16ug.mL-1
MIC=32ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675394
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=8ug.mL-1
MIC>125ug.mL-1
MIC=1ug.mL-1
MIC=0.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675397
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>125ug.mL-1
MIC=63ug.mL-1
MIC=8ug.mL-1
MIC=16ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675396
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=32ug.mL-1
MIC=2ug.mL-1
MIC=0.13ug.mL-1
MIC=0.25ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675398
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=63ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675401
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=32ug.mL-1
MIC=4ug.mL-1
MIC=4ug.mL-1
MIC=63ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675400
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=32ug.mL-1
MIC=32ug.mL-1
MIC=8ug.mL-1
MIC=0.25ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675308
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=8ug.mL-1
MIC=2ug.mL-1
MIC=0.25ug.mL-1
MIC=0.25ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL675402
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=4ug.mL-1
MIC=0.25ug.mL-1
MIC=0.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycolicibacterium smegmatis
External ID: CHEMBL3995600
Protocol: N/A
Comment: Journal: Eur J Med Chem
Year: 2017
Volume: 127
First Page: 223
Last Page: 234
DOI: 10.1016/j.ejmech.2016.12.060

Target ChEMBL ID: CHEMBL613088
ChEMBL Target Name: Mycolicibacterium smegmatis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=105ug.mL-1
MIC=32ug.mL-1
MIC=45ug.mL-1
MIC=32ug.mL-1
MIC=2ug.mL-1
MIC=8ug.mL-1
MIC=512ug.mL-1
MIC=128ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Metallo-beta-lactamase type 2
External ID: CHEMBL1652763
Protocol: N/A
Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Antimicrob. Agents Chemother.
Year: 2009
Volume: 53
Issue: 10
First Page: 4320
Last Page: 4326
DOI: 10.1128/aac.01607-08

Target ChEMBL ID: CHEMBL1667689
ChEMBL Target Name: Metallo-beta-lactamase IND-6
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
PubChem Standard ValueStandard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
60Km=60000nM
Kcat=25/s
145Km=145000nM
Kcat=50/s
13Km=13000nM
KcatNot Determined
KmNot Determined
Kcat=490/s
90Km=90000nM
Kcat=480/s
85Km=85000nM
Kcat=210/s
30Km=30000nM
Kcat=75/s
23Km=23000nM
Kcat>1.2/s
300Km>300000nM
Kcat=115/s
43Km=43000nM
3Km=3000nM
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Metallo-beta-lactamase type 2
External ID: CHEMBL1652764
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2009
Volume: 53
Issue: 10
First Page: 4320
Last Page: 4326
DOI: 10.1128/aac.01607-08

Target ChEMBL ID: CHEMBL1667689
ChEMBL Target Name: Metallo-beta-lactamase IND-6
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
Kcat/Km=1.510'7/M/s
Kcat/Km=6.910'6/M/s
Kcat/Km=1.710'5/M/s
Kcat/Km=3.810'6/M/s
Kcat/KmNot Determined
Kcat/Km=5.410'6/M/s
Kcat/Km=5.610'6/M/s
Kcat/Km=710'6/M/s
Kcat/Km=3.310'6/M/s
Kcat/Km=410'3/M/s
Kcat/Km=2.710'6/M/s
Kcat/Km=6.310'6/M/s
Kcat/Km=2.410'5/M/s
Kcat/Km=2.710'5/M/s
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Metallo-beta-lactamase type 2
External ID: CHEMBL1652765
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2009
Volume: 53
Issue: 10
First Page: 4320
Last Page: 4326
DOI: 10.1128/aac.01607-08

Target ChEMBL ID: CHEMBL1667690
ChEMBL Target Name: IND-like metallo-beta-lactamase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
Kcat/Km=8.410'5/M/s
Kcat/Km=1.510'4/M/s
Kcat/Km=2.410'4/M/s
Kcat/KmNot Determined
Kcat/Km=5.310'4/M/s
Kcat/KmNot Determined
Kcat/Km=3.110'4/M/s
Kcat/KmNot Determined
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Metallo-beta-lactamase type 2
External ID: CHEMBL1652767
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2009
Volume: 53
Issue: 10
First Page: 4320
Last Page: 4326
DOI: 10.1128/aac.01607-08

Target ChEMBL ID: CHEMBL1667692
ChEMBL Target Name: Carbapenem-hydrolyzing beta-lactamase BlaB-1
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
Kcat/Km=2.710'7/M/s
Kcat/Km=1.610'6/M/s
Kcat/Km=7.610'5/M/s
Kcat/Km=210'6/M/s
Kcat/KmNot Determined
Kcat/Km=1.410'5/M/s
Kcat/Km=6.110'6/M/s
Kcat/Km=110'6/M/s
Kcat/Km=210'2/M/s
Kcat/Km=3.910'6/M/s
Kcat/Km=7.910'5/M/s
Kcat/Km=6.610'3/M/s
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL682915
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1980
Volume: 23
Issue: 4
First Page: 405
Last Page: 412
DOI: 10.1021/jm00178a011

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=12.5ug.mL-1
MIC=6.2ug.mL-1
MIC=6.2ug.mL-1
MIC=6.2ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL807842
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>125ug.mL-1
MIC>125ug.mL-1
MIC=32ug.mL-1
MIC=0.25ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL807841
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=8ug.mL-1
MIC>125ug.mL-1
MIC=0.13ug.mL-1
MIC=0.13ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL808006
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=1ug.mL-1
MIC=0.05ug.mL-1
MIC=0.03ug.mL-1
MIC=0.06ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL808005
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=2ug.mL-1
MIC=8ug.mL-1
MIC=16ug.mL-1
MIC=0.13ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL807844
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>125ug.mL-1
MIC>125ug.mL-1
MIC=8ug.mL-1
MIC=32ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL807843
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=4ug.mL-1
MIC=125ug.mL-1
MIC=32ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL3301365
Protocol: N/A
Comment: Data Source: AstraZeneca DMPK/physicochemical
Standard TypeStandard ValueStandard Units
PPB96%
PPB34.42%
PPB87.87%
PPB79.55%
PPB55.73%
PPB99.91%
PPB98.61%
PPB99.81%
PPB87.11%
PPB96.26%
PPB92.32%
PPB66.1%
PPB75.97%
PPB99.19%
PPB62.4%
PPB30.88%
PPB71.99%
PPB98.37%
PPB92.64%
PPB95.72%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Stenotrophomonas maltophilia
External ID: CHEMBL1264475
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2008
Volume: 52
Issue: 3
First Page: 1198
Last Page: 1200
DOI: 10.1128/aac.00682-07

Target ChEMBL ID: CHEMBL612366
ChEMBL Target Name: Stenotrophomonas maltophilia
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>32ug.mL-1
MIC>32ug.mL-1
MIC=16ug.mL-1
MIC=128ug.mL-1
MIC=1024ug.mL-1
MIC=64ug.mL-1
MIC>2048ug.mL-1
MIC=1024ug.mL-1
MIC=4ug.mL-1
MIC=512ug.mL-1
MIC=128ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Stenotrophomonas maltophilia
External ID: CHEMBL1264474
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2008
Volume: 52
Issue: 3
First Page: 1198
Last Page: 1200
DOI: 10.1128/aac.00682-07

Target ChEMBL ID: CHEMBL612366
ChEMBL Target Name: Stenotrophomonas maltophilia
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=0.5ug.mL-1
MIC=8ug.mL-1
MIC>2048ug.mL-1
MIC=128ug.mL-1
MIC=128ug.mL-1
MIC=1024ug.mL-1
MIC>2048ug.mL-1
MIC=1024ug.mL-1
MIC=64ug.mL-1
MIC=256ug.mL-1
MIC=128ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Stenotrophomonas maltophilia
External ID: CHEMBL1264473
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2008
Volume: 52
Issue: 3
First Page: 1198
Last Page: 1200
DOI: 10.1128/aac.00682-07

Target ChEMBL ID: CHEMBL612366
ChEMBL Target Name: Stenotrophomonas maltophilia
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>32ug.mL-1
MIC>32ug.mL-1
MIC>2048ug.mL-1
MIC=256ug.mL-1
MIC=1024ug.mL-1
MIC=1024ug.mL-1
MIC>2048ug.mL-1
MIC=2048ug.mL-1
MIC=64ug.mL-1
MIC=1024ug.mL-1
MIC=256ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL1264778
Protocol: N/A
Comment: Journal: Antimicrob Agents Chemother
Year: 2010
Volume: 54
Issue: 5
First Page: 2219
Last Page: 2224
DOI: 10.1128/aac.00816-09

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=0.5ug.mL-1
MIC=8ug.mL-1
MIC=4ug.mL-1
MIC=32ug.mL-1
MIC=512ug.mL-1
MIC=0.25ug.mL-1
MIC=1ug.mL-1
MIC=128ug.mL-1
MIC=4ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Stenotrophomonas maltophilia
External ID: CHEMBL1264484
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2008
Volume: 52
Issue: 3
First Page: 1198
Last Page: 1200
DOI: 10.1128/aac.00682-07

Target ChEMBL ID: CHEMBL612366
ChEMBL Target Name: Stenotrophomonas maltophilia
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Ratio=5.5
Ratio=0.2
Ratio=3.4
Ratio=0.9
Ratio=2.4
Ratio=1.7
Ratio=3.2
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Stenotrophomonas maltophilia
External ID: CHEMBL1264481
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2008
Volume: 52
Issue: 3
First Page: 1198
Last Page: 1200
DOI: 10.1128/aac.00682-07

Target ChEMBL ID: CHEMBL612366
ChEMBL Target Name: Stenotrophomonas maltophilia
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeActivity Comment
ActivityNot Active
ActivityNot Active
ActivityNot Active
ActivityNot Active
ActivityNot Active
ActivityNot Active
ActivityNot Active
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Stenotrophomonas maltophilia
External ID: CHEMBL1264480
Protocol: N/A
Comment: Journal: Antimicrob. Agents Chemother.
Year: 2008
Volume: 52
Issue: 3
First Page: 1198
Last Page: 1200
DOI: 10.1128/aac.00682-07

Target ChEMBL ID: CHEMBL612366
ChEMBL Target Name: Stenotrophomonas maltophilia
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeActivity Comment
ActivityNot Active
ActivityNot Active
ActivityNot Active
ActivityNot Active
ActivityNot Active
ActivityNot Active
ActivityNot Active
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL1264786
Protocol: N/A
Comment: Journal: Antimicrob Agents Chemother
Year: 2010
Volume: 54
Issue: 5
First Page: 2219
Last Page: 2224
DOI: 10.1128/aac.00816-09

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=8ug.mL-1
MIC=1ug.mL-1
MIC=128ug.mL-1
MIC=2ug.mL-1
MIC=1ug.mL-1
MIC=128ug.mL-1
MIC=8ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Providencia rettgeri
External ID: CHEMBL772076
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 5
First Page: 611
Last Page: 614
DOI: 10.1021/jm00155a004

Target ChEMBL ID: CHEMBL612537
ChEMBL Target Name: Providencia rettgeri
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=0.5ug.mL-1
MIC=0.13ug.mL-1
MIC=0.06ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL1264785
Protocol: N/A
Comment: Journal: Antimicrob Agents Chemother
Year: 2010
Volume: 54
Issue: 5
First Page: 2219
Last Page: 2224
DOI: 10.1128/aac.00816-09

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=8ug.mL-1
MIC=0.5ug.mL-1
MIC=8ug.mL-1
MIC=2ug.mL-1
MIC=64ug.mL-1
MIC=4ug.mL-1
MIC=32ug.mL-1
MIC=32ug.mL-1
MIC=4ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL1264784
Protocol: N/A
Comment: Journal: Antimicrob Agents Chemother
Year: 2010
Volume: 54
Issue: 5
First Page: 2219
Last Page: 2224
DOI: 10.1128/aac.00816-09

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=0.25ug.mL-1
MIC=8ug.mL-1
MIC=16ug.mL-1
MIC=64ug.mL-1
MIC=512ug.mL-1
MIC=2ug.mL-1
MIC=4ug.mL-1
MIC>256ug.mL-1
MIC=64ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL1264783
Protocol: N/A
Comment: Journal: Antimicrob Agents Chemother
Year: 2010
Volume: 54
Issue: 5
First Page: 2219
Last Page: 2224
DOI: 10.1128/aac.00816-09

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC<=0.12ug.mL-1
MIC=1ug.mL-1
MIC=2ug.mL-1
MIC=32ug.mL-1
MIC=128ug.mL-1
MIC=1ug.mL-1
MIC=1ug.mL-1
MIC>256ug.mL-1
MIC=32ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL1264782
Protocol: N/A
Comment: Journal: Antimicrob Agents Chemother
Year: 2010
Volume: 54
Issue: 5
First Page: 2219
Last Page: 2224
DOI: 10.1128/aac.00816-09

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC<=0.12ug.mL-1
MIC<=0.06ug.mL-1
MIC=0.5ug.mL-1
MIC<=0.12ug.mL-1
MIC<=16ug.mL-1
MIC=0.25ug.mL-1
MIC=1ug.mL-1
MIC=0.5ug.mL-1
MIC<=0.12ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL1111862
Protocol: N/A
Comment: Journal: Bioorg Med Chem
Year: 2010
Volume: 18
Issue: 6
First Page: 2123
Last Page: 2130
DOI: 10.1016/j.bmc.2010.02.005

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=50ug.mL-1
MIC=0.3906ug.mL-1
MIC=3.125ug.mL-1
MIC=200ug.mL-1
MIC=0.5ug.mL-1
MIC=0.125ug.mL-1
MIC=8ug.mL-1
MIC=0.03125ug.mL-1
MIC=0.125ug.mL-1
MIC=0.125ug.mL-1
MIC=2ug.mL-1
MIC=128ug.mL-1
MIC=0.0625ug.mL-1
MIC=0.0625ug.mL-1
MIC=8ug.mL-1
MIC=0.0625ug.mL-1
MIC=0.5ug.mL-1
MIC=0.625ug.mL-1
MIC=0.5ug.mL-1
MIC=0.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL1264781
Protocol: N/A
Comment: Journal: Antimicrob Agents Chemother
Year: 2010
Volume: 54
Issue: 5
First Page: 2219
Last Page: 2224
DOI: 10.1128/aac.00816-09

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC<=0.12ug.mL-1
MIC=0.25ug.mL-1
MIC=0.12ug.mL-1
MIC=0.5ug.mL-1
MIC=32ug.mL-1
MIC<=0.12ug.mL-1
MIC<=0.5ug.mL-1
MIC=4ug.mL-1
MIC=0.5ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Pseudomonas aeruginosa
External ID: CHEMBL1264780
Protocol: N/A
Comment: Journal: Antimicrob Agents Chemother
Year: 2010
Volume: 54
Issue: 5
First Page: 2219
Last Page: 2224
DOI: 10.1128/aac.00816-09

Target ChEMBL ID: CHEMBL348
ChEMBL Target Name: Pseudomonas aeruginosa
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC<=0.12ug.mL-1
MIC=0.5ug.mL-1
MIC=2ug.mL-1
MIC=4ug.mL-1
MIC=64ug.mL-1
MIC=0.5ug.mL-1
MIC<=0.5ug.mL-1
MIC=4ug.mL-1
MIC=1ug.mL-1