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462-41-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL2449008
Protocol: N/A
Comment: Journal: Pharm. Res.
Year: 2013
DOI: 10.1007/s11095-013-1232-z
Standard TypeStandard ValueActivity Comment
pKa9Basic pKa
pKa10.6Basic pKa
pKa10.7Basic pKa
pKa10.7Basic pKa
pKa11.1Basic pKa
pKa8.5Basic pKa
pKa9.8Basic pKa
pKa8.9Basic pKa
pKa10.3Basic pKa
pKa11.3Basic pKa
pKa10.1Basic pKa
pKa9.8Basic pKa
pKa10.9Basic pKa
pKa10.2Basic pKa
pKa8.4Basic pKa
pKa9Basic pKa
pKa7.9Basic pKa
pKa9.4Basic pKa
pKa8.8Basic pKa
pKa10.1Basic pKa
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL991844
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 2008
Volume: 51
Issue: 15
First Page: 4359
Last Page: 4369
DOI: 10.1021/jm800219f
Standard TypeStandard RelationStandard Value
pKa=4.62
pKa=4.76
pKa=5.17
pKa=10.7
pKa=4.2
pKa=10.7
pKa=10.7
pKa=4.87
pKa=9.99
pKa=16
pKa=4.85
pKa=11.1
pKa=4.65
pKa=8.9
pKa=9.89
pKa=9.29
pKa=3.58
pKa=3.79
pKa=3.87
pKa=4.14