HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Vitamin D3 receptor

External ID: CHEMBL5164286

Protocol: N/A

Comment: Journal: J Med Chem
Year: 2022
Volume: 65
Issue: 8.0
First Page: 6039
Last Page: 6055
DOI: 10.1021/acs.jmedchem.1c01878

Target ChEMBL ID: CHEMBL1977
ChEMBL Target Name: Vitamin D receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Activity Comment
Activity	NA

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Peroxisome proliferator-activated receptor gamma

External ID: CHEMBL5164289

Protocol: N/A

Comment: Journal: J Med Chem
Year: 2022
Volume: 65
Issue: 8.0
First Page: 6039
Last Page: 6055
DOI: 10.1021/acs.jmedchem.1c01878

Target ChEMBL ID: CHEMBL235
ChEMBL Target Name: Peroxisome proliferator-activated receptor gamma
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Activity Comment
Activity	NA

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL1798350

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2008
Volume: 43
Issue: 4
First Page: 714
Last Page: 740
DOI: 10.1016/j.ejmech.2007.05.007

Standard Type	Standard Relation	Standard Value
LogP	=	0.83
LogP	=	6.169
LogP	=	4.03
LogP	=	6.882
LogP	=	2.14
LogP	=	4.95
LogP	=	3.868
LogP	=	3.354
LogP	=	3.005
LogP	=	2.855
LogP	=	1.994
LogP	=	2.285
LogP	=	0.842
LogP	=	2.481
LogP	=	4.225
LogP	=	3.316
LogP	=	6.036
LogP	=	2.791
LogP	=	2.142
LogP	=	2.81

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Nuclear receptor ROR-alpha

External ID: CHEMBL4827332

Protocol: N/A

Comment: Journal: J Nat Prod
Year: 2021
Volume: 84
Issue: 7.0
First Page: 1882
Last Page: 1888
DOI: 10.1021/acs.jnatprod.0c01276

Target ChEMBL ID: CHEMBL3217403
ChEMBL Target Name: Nuclear receptor ROR-alpha
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Activity Comment
Activity	Not Active
Activity	Active

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Peroxisome proliferator-activated receptor gamma

External ID: CHEMBL5164290

Protocol: N/A

Comment: Journal: J Med Chem
Year: 2022
Volume: 65
Issue: 8.0
First Page: 6039
Last Page: 6055
DOI: 10.1021/acs.jmedchem.1c01878

Target ChEMBL ID: CHEMBL235
ChEMBL Target Name: Peroxisome proliferator-activated receptor gamma
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Activity Comment
Activity	NA

434-16-2 靶点实验数据