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42286-41-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:NAD-dependent protein deacetylase sirtuin-2
External ID: CHEMBL908195
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 2006
Volume: 49
Issue: 26
First Page: 7907
Last Page: 7911
DOI: 10.1021/jm060566j

Target ChEMBL ID: CHEMBL4462
ChEMBL Target Name: NAD-dependent deacetylase sirtuin 2
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
Inhibition=35%
Inhibition=56%
Inhibition=22%
InhibitionNot Determined
Inhibition=21%
Inhibition=27%