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4074-58-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL845877
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2002
Volume: 12
Issue: 2
First Page: 151
Last Page: 154
DOI: 10.1016/s0960-894x(01)00712-0
Standard TypeStandard RelationStandard ValueStandard Units
K1=2576M-1 min-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL845876
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2002
Volume: 12
Issue: 2
First Page: 151
Last Page: 154
DOI: 10.1016/s0960-894x(01)00712-0
Standard TypeStandard RelationStandard ValueStandard Units
K1=928M-1 min-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:CCRF-HSB-2
External ID: CHEMBL929830
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem.
Year: 2008
Volume: 16
Issue: 2
First Page: 922
Last Page: 940
DOI: 10.1016/j.bmc.2007.10.014

Target ChEMBL ID: CHEMBL614541
ChEMBL Target Name: CCRF-HSB-2
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
IC50=0.047ug.mL-1
IC50=1.8ug.mL-1
IC50=1.57ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:KB
External ID: CHEMBL929831
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem.
Year: 2008
Volume: 16
Issue: 2
First Page: 922
Last Page: 940
DOI: 10.1016/j.bmc.2007.10.014

Target ChEMBL ID: CHEMBL398
ChEMBL Target Name: KB
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsData Validity Comment
IC50=0.23ug.mL-1
IC50=2.1ug.mL-1
IC50=1.89ug.mL-1