HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL632012

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat/Km	=	53	M-1 s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL632013

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat/Km	=	29.1	M-1 s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL632014

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat/Km	=	1.4	M-1 s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL629622

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat/Km	=	5.9	M-1 s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL628505

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Units	Activity Comment
Km	nM	Not Determined

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL629623

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat/Km	=	10.1	M-1 s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL629624

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat/Km	=	0.6	M-1 s-1
k cat/Km	=	39	M-1 s-1
k cat/Km	=	6	M-1 s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL850875

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value
Ratio	=	32
Ratio	=	48
Ratio	=	38

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL628506

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Units	Activity Comment
Km	nM	Not Determined

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL628507

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Units	Activity Comment
Km	nM	Not Determined

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL629626

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat/Kuncat	=	18000	M-1 s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL629627

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat/Kuncat	=	6300	M-1 s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL857742

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Activity Comment
k cat	Not Determined

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL631490

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat	=	350	s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL631491

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Activity Comment
k cat	Not Determined

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL631492

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Activity Comment
k cat	Not Determined

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL631493

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
k cat	=	220	s-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL857732

Protocol: N/A

Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1997
Volume: 7
Issue: 19
First Page: 2497
Last Page: 2502
DOI: 10.1016/S0960-894X(97)10003-8

Standard Type	Standard Relation	Standard Value	Standard Units
K amine	=	0.0185	M-1 s-1
K amine	=	0.82	M-1 s-1
K amine	=	0.16	M-1 s-1

39835-28-4 靶点实验数据