HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Histone acetyltransferase p300

External ID: CHEMBL3269130

Protocol: N/A

Comment: Journal: Eur. J. Med. Chem.
Year: 2014
Volume: 80
First Page: 569
Last Page: 578
DOI: 10.1016/j.ejmech.2014.04.042

Target ChEMBL ID: CHEMBL3784
ChEMBL Target Name: Histone acetyltransferase p300
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	4	%
Inhibition	=	34	%
Inhibition	=	27	%
Inhibition	=	31	%
Inhibition	=	21	%
Inhibition	=	14	%
Inhibition	=	26	%
Inhibition	=	36	%
Inhibition	=	16	%
Inhibition	=	22	%
Inhibition	=	42	%
Inhibition	=	32	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Histone acetyltransferase KAT2B

External ID: CHEMBL3269133

Protocol: N/A

Comment: Journal: Eur. J. Med. Chem.
Year: 2014
Volume: 80
First Page: 569
Last Page: 578
DOI: 10.1016/j.ejmech.2014.04.042

Target ChEMBL ID: CHEMBL5500
ChEMBL Target Name: Histone acetyltransferase PCAF
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	3	%
Inhibition	=	1	%
Inhibition	=	0	%
Inhibition	=	0	%
Inhibition	=	5	%
Inhibition	=	0	%
Inhibition	=	5	%
Inhibition	=	10	%
Inhibition	=	7	%
Inhibition	=	0	%
Inhibition	=	13	%
Inhibition	=	12	%

36941-40-9 靶点实验数据