HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Methionine aminopeptidase 2

External ID: CHEMBL872187

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: J. Med. Chem.
Year: 2005
Volume: 48
Issue: 18
First Page: 5644
Last Page: 5647
DOI: 10.1021/jm050408c

Target ChEMBL ID: CHEMBL3922
ChEMBL Target Name: Methionine aminopeptidase 2
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units
0.112	Ki	=	112	nM
0.15	Ki	=	150	nM
0.03	Ki	=	30	nM
1	Ki	>	1000	nM
0.337	Ki	=	337	nM
0.003	Ki	=	3	nM
0.001	Ki	=	1	nM
0.3	Ki	=	300	nM
0.28	Ki	=	280	nM
0.016	Ki	=	16	nM
0.004	Ki	=	4	nM
0.041	Ki	=	41	nM
0.006	Ki	=	6	nM
0.26	Ki	=	260	nM
1	Ki	>	1000	nM
0.006	Ki	=	6	nM
0.003	Ki	=	3	nM
0.008	Ki	=	8	nM
0.018	Ki	=	18	nM
0.013	Ki	=	13	nM

369363-75-7 靶点实验数据