前往化源商城

36357-32-1 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Candida albicans
External ID: CHEMBL3796409
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 10
First Page: 2438
Last Page: 2441
DOI: 10.1016/j.bmcl.2016.03.115

Target ChEMBL ID: CHEMBL366
ChEMBL Target Name: Candida albicans
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Saccharomyces cerevisiae
External ID: CHEMBL3796408
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 10
First Page: 2438
Last Page: 2441
DOI: 10.1016/j.bmcl.2016.03.115

Target ChEMBL ID: CHEMBL361
ChEMBL Target Name: Saccharomyces cerevisiae
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:J774.A1
External ID: CHEMBL2025507
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2012
Volume: 22
Issue: 9
First Page: 3177
Last Page: 3180
DOI: 10.1016/j.bmcl.2012.03.045

Target ChEMBL ID: CHEMBL614040
ChEMBL Target Name: J774.A1
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
FC=1.86
FC=2.05
FC=3.09
FC=1.47
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL3796407
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 10
First Page: 2438
Last Page: 2441
DOI: 10.1016/j.bmcl.2016.03.115

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Bacillus spizizenii
External ID: CHEMBL3796406
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 10
First Page: 2438
Last Page: 2441
DOI: 10.1016/j.bmcl.2016.03.115

Target ChEMBL ID: CHEMBL613907
ChEMBL Target Name: Bacillus spizizenii
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Candida albicans
External ID: CHEMBL3796411
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 10
First Page: 2438
Last Page: 2441
DOI: 10.1016/j.bmcl.2016.03.115

Target ChEMBL ID: CHEMBL366
ChEMBL Target Name: Candida albicans
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MFC99.9>200ug ml-1
MFC99.9>200ug ml-1
MFC99.9>200ug ml-1
MFC99.9>200ug ml-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Artemia salina
External ID: CHEMBL3050935
Protocol: N/A
Comment: Journal: J Agric Food Chem
Year: 2012
Volume: 60
Issue: 13
First Page: 3424
Last Page: 3431
DOI: 10.1021/jf300146n

Target ChEMBL ID: CHEMBL612341
ChEMBL Target Name: Artemia salina
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
LC50>100ug.mL-1
LC50=44.8ug.mL-1
LC50>100ug.mL-1
LC50>100ug.mL-1
LC50=40.5ug.mL-1
LC50=52.7ug.mL-1
LC50>100ug.mL-1
LC50=73.7ug.mL-1
LC50<1ug.mL-1
LC50>100ug.mL-1
LC50=66.1ug.mL-1
LC50=83.7ug.mL-1
LC50>100ug.mL-1
LC50>100ug.mL-1
LC50>100ug.mL-1
LC50>100ug.mL-1
LC50>100ug.mL-1
LC50>100ug.mL-1
LC50=73.2ug.mL-1
LC50=80.8ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Saccharomyces cerevisiae
External ID: CHEMBL3796410
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 10
First Page: 2438
Last Page: 2441
DOI: 10.1016/j.bmcl.2016.03.115

Target ChEMBL ID: CHEMBL361
ChEMBL Target Name: Saccharomyces cerevisiae
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MFC99.9>200ug ml-1
MFC99.9>200ug ml-1
MFC99.9>200ug ml-1
MFC99.9>200ug ml-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:J774.A1
External ID: CHEMBL2025505
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2012
Volume: 22
Issue: 9
First Page: 3177
Last Page: 3180
DOI: 10.1016/j.bmcl.2012.03.045

Target ChEMBL ID: CHEMBL614040
ChEMBL Target Name: J774.A1
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueActivity Comment
FC=1.29
FC=1.54
FC=1.65
FC=1.56
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL3796405
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 10
First Page: 2438
Last Page: 2441
DOI: 10.1016/j.bmcl.2016.03.115

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
MIC>200ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:J774.A1
External ID: CHEMBL2025506
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2012
Volume: 22
Issue: 9
First Page: 3177
Last Page: 3180
DOI: 10.1016/j.bmcl.2012.03.045

Target ChEMBL ID: CHEMBL614040
ChEMBL Target Name: J774.A1
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
FC=3.5
FC=1.62
FC=4.49
FC=1.36